| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4605643 | B | Inhibition of human ABL1 assessed as residual activity using EAIYAAPFAKKK as substrate by [gamma-33P]-ATP assay | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 2. | ALA4605644 | A | Cytotoxicity against HEK293 cells assessed as reduction in cell viability incubated for 72 hrs by Cell Titer Glo 2.0 reagent based assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 3. | ALA4605645 | A | Metabolic stability in human liver microsomes assessed as half life at 3 uM measured up to 30 mins in presence of NADPH by LS-MS/MS analysis | Homo sapiens | 5 | microsome format | Scientific Literature | ||
| 4. | ALA4605646 | A | Cytotoxicity against human THLE3 assessed as reduction in cell viability incubated for 72 hrs by Cell Titer Glo 2.0 reagent based assay | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 5. | ALA4605647 | A | Metabolic stability in mouse liver microsomes assessed as half life at 3 uM measured up to 30 mins in presence of NADPH by LS-MS/MS analysis | Mus musculus | 5 | microsome format | Scientific Literature | ||
| 6. | ALA4605648 | A | Inhibition of human recombinant CYP3A4 expressed in insect cell microsomes in presence of NADPH by fluorescence assay | Homo sapiens | 8 | microsome format | Scientific Literature | ||
| 7. | ALA4605649 | B | Inhibition of human ERG incubated for 4 hrs by competitive fluorescence tracer binding based assay | Homo sapiens | 8 | single protein format | Scientific Literature | ||
| 8. | ALA4605650 | B | Inhibition of ABL1 (unknown origin) assessed as residual activity at 10 uM incubated for 5 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 9. | ALA4605651 | B | Inhibition of DDR2 (unknown origin) assessed as residual activity at 10 uM incubated for 5 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 10. | ALA4605652 | B | Inhibition of PDGFRalpha (unknown origin) assessed as residual activity at 10 uM incubated for 5 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 11. | ALA4605653 | B | Inhibition of SRC (unknown origin) assessed as residual activity at 10 uM incubated for 5 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 12. | ALA4605654 | B | Inhibition of EPHB2 (unknown origin) assessed as residual activity at 10 uM incubated for 5 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 13. | ALA4605655 | B | Inhibition of EPHB3 (unknown origin) assessed as residual activity at 10 uM incubated for 5 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 14. | ALA4605656 | B | Inhibition of LCK (unknown origin) assessed as residual activity at 10 uM incubated for 5 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 15. | ALA4605657 | B | Inhibition of EPHB4 (unknown origin) assessed as residual activity at 10 uM incubated for 5 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 16. | ALA4605658 | B | Inhibition of NEK6 (unknown origin) assessed as residual activity at 10 uM incubated for 5 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 17. | ALA4605659 | B | Inhibition of VEGFR (unknown origin) assessed as residual activity at 10 uM incubated for 5 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 18. | ALA4605660 | B | Inhibition of MAP4K3 (unknown origin) assessed as residual activity at 10 uM incubated for 5 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 19. | ALA4605661 | B | Inhibition of ABL1 (unknown origin) assessed as residual activity incubated for 5 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 20. | ALA4605662 | B | Inhibition of DDR2 (unknown origin) assessed as residual activity incubated for 5 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay | Homo sapiens | 2 | single protein format | Scientific Literature |
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