| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4619369 | Binding | Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET method | Homo sapiens | 39 | ALA4616719 | single protein format | Scientific Literature | |
| 2. | ALA4619370 | ADME | Half life in C57BL/6N mouse at 2 mg/kg, po after 0.5 to 8 hrs by LC-MS/MS analysis | Mus musculus | 4 | ALA4616719 | organism-based format | Scientific Literature | |
| 3. | ALA4619371 | ADME | Tmax in C57BL/6N mouse at 2 mg/kg, po after 0.5 to 8 hrs by LC-MS/MS analysis | Mus musculus | 4 | ALA4616719 | organism-based format | Scientific Literature | |
| 4. | ALA4619372 | ADME | Cmax in C57BL/6N mouse at 2 mg/kg, po after 0.5 to 8 hrs by LC-MS/MS analysis | Mus musculus | 4 | ALA4616719 | organism-based format | Scientific Literature | |
| 5. | ALA4619373 | ADME | AUClast in C57BL/6N mouse at 2 mg/kg, po after 0.5 to 8 hrs by LC-MS/MS analysis | Mus musculus | 4 | ALA4616719 | organism-based format | Scientific Literature | |
| 6. | ALA4619374 | ADME | Permeability in MDCK cells | Canis lupus familiaris | 1 | ALA4616719 | cell-based format | Scientific Literature | |
| 7. | ALA4619375 | ADME | Protein binding in mouse plasma | Mus musculus | 2 | ALA4616719 | cell-free format | Scientific Literature | |
| 8. | ALA4619376 | Binding | Inhibition of PKCzeta in human THP1 cells assessed as reduction in LPS-induced TNFalpha production pre-incubated for 60 mins before LPS simulations for 4 hrs by HTRF assay | Homo sapiens | 2 | ALA4616719 | cell-based format | Scientific Literature | |
| 9. | ALA5127341 | Binding | Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFKC as substrate measured by TR-FRET assay | Homo sapiens | 6 | ALA5126516 | single protein format | Scientific Literature |
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