| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4629361 | Binding | Reversible inhibition of human MAGL L179S/L186S mutant using 4-methylumbelliferyl butyrate as substrate measured after 5 mins by fluorescence assay | Homo sapiens | 17 | ALA4627378 | assay format | Scientific Literature | |
| 2. | ALA4629362 | Binding | Inhibition of MAGL in rat brain homogenate assessed as accumulation of 2-AG at 10 uM measured after 15 mins by HPLC-MS analysis relative to control | Rattus norvegicus | 9 | ALA4627378 | tissue-based format | Scientific Literature | |
| 3. | ALA4629364 | ADME | Drug concentration in plasma of rat at 10 mg/kg, po | Rattus norvegicus | 4 | ALA4627378 | organism-based format | Scientific Literature | |
| 4. | ALA4629365 | ADME | Drug concentration in brain of rat at 10 mg/kg, po | Rattus norvegicus | 4 | ALA4627378 | organism-based format | Scientific Literature | |
| 5. | ALA4629366 | ADME | Ratio of drug concentration in brain to plasma of rat | Rattus norvegicus | 4 | ALA4627378 | cell-free format | Scientific Literature | |
| 6. | ALA4629367 | Binding | Inhibition of MAGL in rat brain homogenate assessed as accumulation of 2-AG at 1 uM measured after 15 mins by HPLC-MS analysis relative to control | Rattus norvegicus | 12 | ALA4627378 | tissue-based format | Scientific Literature |
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