# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4620599 | Binding | Inhibition of human CDK2/Cyclin A assessed as residual activity at 1 uM using Histone 1 as substrate in presence of ATP incubated for 50 mins by ADP-GloTM assay relative to control | Homo sapiens | 13 | ALA4619742 | protein complex format | Scientific Literature | |
2. | ALA4620600 | Binding | Inhibition of human recombinant CDK5/p25 expressed in bacteria assessed as residual activity at 1 uM using Histone 1 as substrate in presence of ATP incubated for 50 mins by ADP-GloTM assay relative to control | Homo sapiens | 13 | ALA4619742 | assay format | Scientific Literature | |
3. | ALA4620601 | Binding | Inhibition of human recombinant CDK9/Cyclin T expressed in baculovirus in Sf9 insect cells assessed as residual activity at 1 uM using SPTSPSYSPTSPSYSPTSPSKKKK as substrate in presence of ATP incubated for 50 mins by ADP-GloTM assay relative to control | Homo sapiens | 13 | ALA4619742 | cell-based format | Scientific Literature | |
4. | ALA4620602 | Binding | Inhibition of human recombinant Haspin (470 to 798 residues) expressed in bacteria assessed as residual activity at 1 uM using Histone H3 and ARTKQTARKSTGGKAPRKQLA as substrate in presence of ATP incubated for 50 mins by ADP-GloTM assay relative to control | Homo sapiens | 13 | ALA4619742 | assay format | Scientific Literature | |
5. | ALA4620603 | Binding | Inhibition of human recombinant PIM1 expressed in bacteria assessed as residual activity at 1 uM using Histone 1 as substrate in presence of ATP incubated for 50 mins by ADP-GloTM assay relative to control | Homo sapiens | 13 | ALA4619742 | assay format | Scientific Literature | |
6. | ALA4620604 | Binding | Inhibition of porcine CK1-delta assessed as residual activity at 1 uM using RRKHAAIGSpAYSITA as substrate in presence of ATP incubated for 50 mins by ADP-GloTM assay relative to control | Sus scrofa domesticus | 13 | ALA4619742 | single protein format | Scientific Literature | |
7. | ALA4620605 | Binding | Inhibition of porcine GSK3-alpha/GSK3-Beta assessed as residual activity at 1 uM using RAAVPPSPSLSRHSSPHQSpEDEEE as substrate in presence of ATP incubated for 50 mins by ADP-GloTM assay relative to control | Sus scrofa domesticus | 13 | ALA4619742 | protein format | Scientific Literature | |
8. | ALA4620606 | Binding | Inhibition of human recombinant CDK9/Cyclin T expressed in baculovirus in Sf9 insect cells using SPTSPSYSPTSPSYSPTSPSKKKK as substrate in presence of ATP incubated for 50 mins by ADP-GloTM assay | Homo sapiens | 2 | ALA4619742 | cell-based format | Scientific Literature | |
9. | ALA4620607 | Binding | Inhibition of leishmania major CK1 at 1 uM using RRKHAAIGSpAYSIT as substrate in presence of ATP incubated for 50 mins by ADP-GloTM assay relative to control | Leishmania major | 13 | ALA4619742 | assay format | Scientific Literature | |
10. | ALA4620608 | Binding | Inhibition of human recombinant Haspin (470 to 798 residues) expressed in bacteria using Histone H3 and ARTKQTARKSTGGKAPRKQLA as substrate in presence of ATP incubated for 50 mins by ADP-GloTM assay | Homo sapiens | 4 | ALA4619742 | assay format | Scientific Literature |