| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4737600 | B | Inhibition of recombinant human PI3Kalpha using PIP2 as substrate incubated for 1 hr by kinase-glo luminescent assay | Homo sapiens | 8 | ALA4732196 | single protein format | Scientific Literature | |
| 2. | ALA4737601 | B | Inhibition of recombinant human N-terminal FLAG-tagged mTOR (1362 to end amino acids) using ULight-4E-BP1 as substrate incubated for 1 hr by LANCE Ultra assay | Homo sapiens | 8 | ALA4732196 | single protein format | Scientific Literature | |
| 3. | ALA4737602 | F | Growth inhibition of human PC3 cells after 72 hrs by sulforhodamine B assay | Homo sapiens | 8 | ALA4732196 | cell-based format | Scientific Literature | |
| 4. | ALA4737603 | F | Growth inhibition of human U87MG cells after 72 hrs by sulforhodamine B assay | Homo sapiens | 8 | ALA4732196 | cell-based format | Scientific Literature | |
| 5. | ALA4737604 | B | Inhibition of PI3Kbeta (unknown origin) using PIP2 as substrate measured after 1 hr by ADP-glo assay | Homo sapiens | 2 | ALA4732196 | single protein format | Scientific Literature | |
| 6. | ALA4737605 | B | Inhibition of recombinant human full-length His-tagged PI3Kgamma expressed in baculovirus expression system using PIP2 as substrate measured after 1 hr by ADP-glo assay | Homo sapiens | 2 | ALA4732196 | assay format | Scientific Literature | |
| 7. | ALA4737606 | B | Inhibition of PI3Kdelta (unknown origin) using PIP2 as substrate measured after 1 hr by ADP-glo assay | Homo sapiens | 2 | ALA4732196 | single protein format | Scientific Literature | |
| 8. | ALA4737607 | B | Inhibition of human partial length AAK1 (G25 to L333 residues) expressed in bacterial system assessed as residual activity at 10 uM by kinome scan method relative to control | Homo sapiens | 1 | ALA4732196 | assay format | Scientific Literature | |
| 9. | ALA4737608 | B | Inhibition of human partial length ACVR2A (V171 to T499 residues) expressed in bacterial system assessed as residual activity at 10 uM by kinome scan method relative to control | Homo sapiens | 1 | ALA4732196 | assay format | Scientific Literature | |
| 10. | ALA4737609 | B | Inhibition of human partial length ACVR2B (H169 to D504 residues) expressed in bacterial system assessed as residual activity at 10 uM by kinome scan method relative to control | Homo sapiens | 1 | ALA4732196 | assay format | Scientific Literature | |
| 11. | ALA4737610 | B | Inhibition of human partial length ANKK1 (M1 to A305 residues) expressed in bacterial system assessed as residual activity at 10 uM by kinome scan method relative to control | Homo sapiens | 1 | ALA4732196 | assay format | Scientific Literature | |
| 12. | ALA4737611 | B | Inhibition of human partial length BIKE (S34 to N329 residues) expressed in bacterial system assessed as residual activity at 10 uM by kinome scan method relative to control | Homo sapiens | 1 | ALA4732196 | assay format | Scientific Literature | |
| 13. | ALA4737612 | B | Inhibition of human partial length BUB1 (Q724 to K1085 residues) expressed in bacterial system assessed as residual activity at 10 uM by kinome scan method relative to control | Homo sapiens | 1 | ALA4732196 | assay format | Scientific Literature | |
| 14. | ALA4737613 | B | Inhibition of human partial length CDC2L1 (P353 to G692 residues) expressed in bacterial system assessed as residual activity at 10 uM by kinome scan method relative to control | Homo sapiens | 1 | ALA4732196 | assay format | Scientific Literature | |
| 15. | ALA4737614 | B | Inhibition of human partial length CDK11 (M1 to N360 residues) expressed in bacterial system assessed as residual activity at 10 uM by kinome scan method relative to control | Homo sapiens | 1 | ALA4732196 | assay format | Scientific Literature | |
| 16. | ALA4737615 | B | Inhibition of human partial length CDK8 (M1 to T360 residues) expressed in bacterial system assessed as residual activity at 10 uM by kinome scan method relative to control | Homo sapiens | 1 | ALA4732196 | assay format | Scientific Literature | |
| 17. | ALA4737616 | B | Inhibition of human partial length CDKL1 (M1 to I358 residues) expressed in bacterial system assessed as residual activity at 10 uM by kinome scan method relative to control | Homo sapiens | 1 | ALA4732196 | assay format | Scientific Literature | |
| 18. | ALA4737617 | B | Inhibition of human partial length CDKL1 (M1 to D327 residues) expressed in bacterial system assessed as residual activity at 10 uM by kinome scan method relative to control | Homo sapiens | 1 | ALA4732196 | assay format | Scientific Literature | |
| 19. | ALA4737618 | B | Inhibition of human partial length CDKL5 (M1 to S337 residues) expressed in mammalian expression system assessed as residual activity at 10 uM by kinome scan method relative to control | Homo sapiens | 1 | ALA4732196 | assay format | Scientific Literature | |
| 20. | ALA4737619 | B | Inhibition of human partial length CIT (M68 to E432 residues) expressed in bacterial expression system assessed as residual activity at 10 uM by kinome scan method relative to control | Homo sapiens | 1 | ALA4732196 | assay format | Scientific Literature |
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