# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4670288 | B | Inhibition of human TREK1 in open state expressed in CHO cells in presence of 10 uM TREK1 activator arachidonic acid by whole-cell patch-clamp electrophysiological method | Homo sapiens | 1 | ALA4665784 | cell-based format | Scientific Literature | |
2. | ALA4670289 | B | Inhibition of human TREK1 R207A mutant at intermediate transition state expressed in CHO cells by whole-cell patch-clamp electrophysiological method | Homo sapiens | 2 | ALA4665784 | cell-based format | Scientific Literature | |
3. | ALA4670290 | B | Inhibition of human TRAAK at intermediate transition state expressed in CHO cells by whole-cell patch-clamp electrophysiological method | Homo sapiens | 1 | ALA4665784 | cell-based format | Scientific Literature | |
4. | ALA4670291 | B | Inhibition of human TREK2 at intermediate transition state expressed in CHO cells by whole-cell patch-clamp electrophysiological method | Homo sapiens | 1 | ALA4665784 | cell-based format | Scientific Literature | |
5. | ALA4670292 | B | Inhibition of human TREK1 D294A mutant at intermediate transition state expressed in CHO cells by whole-cell patch-clamp electrophysiological method | Homo sapiens | 3 | ALA4665784 | cell-based format | Scientific Literature | |
6. | ALA4670293 | B | Inhibition of human TREK1 S290A mutant at intermediate transition state expressed in CHO cells by whole-cell patch-clamp electrophysiological method | Homo sapiens | 3 | ALA4665784 | cell-based format | Scientific Literature | |
7. | ALA4670294 | B | Inhibition of human TREK1 V288A mutant at intermediate transition state expressed in CHO cells by whole-cell patch-clamp electrophysiological method | Homo sapiens | 1 | ALA4665784 | cell-based format | Scientific Literature | |
8. | ALA4670295 | B | Inhibition of human TREK1 W295A mutant at intermediate transition state expressed in CHO cells by whole-cell patch-clamp electrophysiological method | Homo sapiens | 1 | ALA4665784 | cell-based format | Scientific Literature | |
9. | ALA4670296 | B | Inhibition of human TREK1 M291A mutant at intermediate transition state expressed in CHO cells by whole-cell patch-clamp electrophysiological method | Homo sapiens | 1 | ALA4665784 | cell-based format | Scientific Literature | |
10. | ALA4670297 | B | Inhibition of human TREK1 T211A mutant at intermediate transition state expressed in CHO cells by whole-cell patch-clamp electrophysiological method | Homo sapiens | 1 | ALA4665784 | cell-based format | Scientific Literature | |
11. | ALA4670298 | B | Inhibition of human TREK1 at intermediate transition state expressed in CHO cells assessed as decrease in probability of TREK1 channel being in open state by single-channel recordings based by inside-out patch method | Homo sapiens | 1 | ALA4665784 | cell-based format | Scientific Literature | |
12. | ALA4670299 | B | Effect on channel conductance of human TREK1 expressed in CHO cells by single-channel recordings based by inside-out patch method | Homo sapiens | 1 | ALA4665784 | cell-based format | Scientific Literature | |
13. | ALA4670300 | B | Inhibition of human TREK1 at intermediate transition state expressed in CHO cells by whole-cell patch-clamp electrophysiological method | Homo sapiens | 3 | ALA4665784 | cell-based format | Scientific Literature |