| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4714156 | B | Displacement of [3H]-gabapentin from human Cav alpha2delta1 expressed in CHO-K1 cell membranes incubated for 60 mins by scintillation counting method | Homo sapiens | 39 | ALA4706691 | cell membrane format | Scientific Literature | |
| 2. | ALA4714158 | B | Displacement of [3H]-nisoxetine from human NET expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting method | Homo sapiens | 39 | ALA4706691 | cell membrane format | Scientific Literature | |
| 3. | ALA4714159 | B | Inhibition of human NET expressed in HEK293 cells assessed as reduction in ASP+ uptake incubated for 20 mins before ASP+ addition and measured after 90 mins by scintillation counting method | Homo sapiens | 39 | ALA4706691 | cell-based format | Scientific Literature | |
| 4. | ALA4714161 | A | Intrinsic clearance in human liver microsomes | Homo sapiens | 3 | ALA4706691 | microsome format | Scientific Literature | |
| 5. | ALA4714162 | A | Intrinsic clearance in rat liver microsomes | Rattus norvegicus | 3 | ALA4706691 | microsome format | Scientific Literature | |
| 6. | ALA4714163 | A | Inhibition of human CYP1A2 at 1 uM relative to control | Homo sapiens | 3 | ALA4706691 | single protein format | Scientific Literature | |
| 7. | ALA4714164 | A | Inhibition of human CYP2C9 at 1 uM relative to control | Homo sapiens | 3 | ALA4706691 | single protein format | Scientific Literature | |
| 8. | ALA4714165 | A | Inhibition of human CYP2C19 at 1 uM relative to control | Homo sapiens | 3 | ALA4706691 | single protein format | Scientific Literature | |
| 9. | ALA4714166 | A | Inhibition of human CYP2D6 at 1 uM relative to control | Homo sapiens | 3 | ALA4706691 | single protein format | Scientific Literature | |
| 10. | ALA4714167 | A | Inhibition of human CYP3A4 at 1 uM relative to control | Homo sapiens | 3 | ALA4706691 | single protein format | Scientific Literature | |
| 11. | ALA4714168 | B | Inhibition of human ERG | Homo sapiens | 3 | ALA4706691 | single protein format | Scientific Literature | |
| 12. | ALA4714169 | P | Kinetic solubility of the compound | 2 | ALA4706691 | small-molecule physicochemical format | Scientific Literature | ||
| 13. | ALA4714170 | A | Intrinsic clearance in mouse liver microsomes | Mus musculus | 2 | ALA4706691 | microsome format | Scientific Literature | |
| 14. | ALA5228412 | B | Inhibition of NET (unknown origin) | Homo sapiens | 1 | ALA5226328 | single protein format | Scientific Literature | |
| 15. | ALA5228419 | B | Binding affinity to calcium channel alpha2delta1 (unknown origin) | Homo sapiens | 2 | ALA5226328 | single protein format | Scientific Literature |
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