| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4672965 | B | Protac binding affinity at CRBN/BCR-ABL (unknown origin) assessed as binding to phosphorylated c-ABL kinase domain by Kinomescan assay | Homo sapiens | 5 | protein format | Scientific Literature | ||
| 2. | ALA4672966 | B | Protac binding affinity at CRBN/BCR-ABL (unknown origin) assessed as binding to non phosphorylated c-ABL kinase domain by Kinomescan assay | Homo sapiens | 5 | protein format | Scientific Literature | ||
| 3. | ALA4672967 | B | Protac activity at CRBN/BCR-ABL in human K562 cells assessed as induction of BCR-ABL degradation at 2.5 uM incubated for 24 hrs by western blot analysis relative to control | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 4. | ALA4672968 | B | Protac activity at CRBN/BCR-ABL in human K562 cells assessed as induction of BCR-ABL degradation at 1 uM incubated for 24 hrs by western blot analysis relative to control | Homo sapiens | 5 | cell-based format | Scientific Literature |
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