# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4714732 | B | Inhibition of recombinant human full-length His-tagged TAK1-TAB1 fusion protein (437 to 504 residues) expressed in baculovirus expression system using fluorescein-MAP2K1 as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins in presence of ATP by lanthascreen TR-FRET assay | Homo sapiens | 44 | ALA4706727 | assay format | Scientific Literature | |
2. | ALA4714745 | B | Inhibition of wild-type human full length CSNK2A1 (M1 to Q391 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4706727 | assay format | Scientific Literature | |
3. | ALA4714746 | B | Inhibition of wild-type human full length CSNK2A2 (M1 to R350 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4706727 | assay format | Scientific Literature | |
4. | ALA4714747 | B | Inhibition of human partial length FLT3 D835V mutant (V592 to Y969 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4706727 | assay format | Scientific Literature | |
5. | ALA4714748 | B | Inhibition of wild-type Plasmodium falciparum 3D7 full-length CDPK1 (M1 to S524 residues) expressed in mammalian expression system at 10 uM by kinomescan method relative to control | Plasmodium falciparum 3D7 | 1 | ALA4706727 | assay format | Scientific Literature | |
6. | ALA4714750 | B | Inhibition of wild-type human partial length PIK3CD (R108 to Q1044 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4706727 | assay format | Scientific Literature | |
7. | ALA4714751 | B | Inhibition wild type human partial length PIP5K1C (M1 to T668 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4706727 | assay format | Scientific Literature |