# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4729760 | F | Inhibition glucose production in C57BLKS mouse primary hepatocytes at 100 uM after 4 hrs by colorimetric glucose assay | Mus musculus | 2 | cell-based format | Scientific Literature | ||
2. | ALA4729761 | B | Inhibition of human wild type FBPase expressed in Escherichia coli BL12 (DE3) by malachite green method | Homo sapiens | 36 | assay format | Scientific Literature | ||
3. | ALA4729762 | B | Inhibition of wild type human FBPase | Homo sapiens | 1 | single protein format | Scientific Literature | ||
4. | ALA4729763 | B | Inhibition of human FBPase C1285 mutant | Homo sapiens | 1 | assay format | Scientific Literature | ||
5. | ALA4729764 | B | Inhibition of human FBPase S124A mutant | Homo sapiens | 1 | single protein format | Scientific Literature | ||
6. | ALA4729765 | B | Inhibition of human FBPase N125A mutant | Homo sapiens | 1 | single protein format | Scientific Literature | ||
7. | ALA4729766 | B | Inhibition of human FBPase D127A mutant | Homo sapiens | 1 | single protein format | Scientific Literature | ||
8. | ALA4729767 | B | Inhibition of human FBPase R243A mutant | Homo sapiens | 1 | single protein format | Scientific Literature | ||
9. | ALA4729768 | B | Inhibition of human FBPase R254A mutant | Homo sapiens | 1 | assay format | Scientific Literature | ||
10. | ALA4729769 | B | Inhibition of human FBPase Y258A mutant | Homo sapiens | 1 | single protein format | Scientific Literature | ||
11. | ALA4729770 | B | Selectivity ratio of IC50 for human FBPase C1285 mutant to IC50 for human wild type FBPase | Homo sapiens | 1 | assay format | Scientific Literature | ||
12. | ALA4729771 | B | Selectivity ratio of IC50 for human FBPase S124A mutant to IC50 for human wild type FBPase | Homo sapiens | 1 | assay format | Scientific Literature | ||
13. | ALA4729772 | B | Selectivity ratio of IC50 for human FBPase N125A mutant to IC50 for human wild type FBPase | Homo sapiens | 1 | assay format | Scientific Literature | ||
14. | ALA4729773 | B | Selectivity ratio of IC50 for human FBPase D127A mutant to IC50 for human wild type FBPase | Homo sapiens | 1 | assay format | Scientific Literature | ||
15. | ALA4729774 | B | Selectivity ratio of IC50 for human FBPase R243A mutant to IC50 for human wild type FBPase | Homo sapiens | 1 | assay format | Scientific Literature | ||
16. | ALA4729775 | B | Selectivity ratio of IC50 for human FBPase R254A mutant to IC50 for human wild type FBPase | Homo sapiens | 1 | assay format | Scientific Literature | ||
17. | ALA4729776 | B | Selectivity ratio of IC50 for human FBPase Y258A mutant to IC50 for human wild type FBPase | Homo sapiens | 1 | assay format | Scientific Literature |