| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4672124 | Binding | Inhibition of KEAP1 interaction with Nrf2 in human SH-SY5Y cells transfected with NeH2-LUC assessed as activation of Nrf2 signaling pathway measured after 18 hrs by bright-Glo luciferase assay | Homo sapiens | 34 | ALA4665857 | cell-based format | Scientific Literature | |
| 2. | ALA4672125 | Binding | Inhibition of KEAP1 interaction with Nrf2 in human SH-SY5Y. cells transfected with ARE-LUC assessed as activation of Nrf2 signaling pathway measured after 18 hrs by bright-Glo luciferase assay | Homo sapiens | 34 | ALA4665857 | cell-based format | Scientific Literature | |
| 3. | ALA4672126 | Binding | Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assay | Homo sapiens | 72 | ALA4665857 | single protein format | Scientific Literature |
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