| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4715191 | F | Antagonist activity in CXCR2 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization pretreated with Fluo-4AM for 45 mins followed by compound addition and measured after 10 mins by Fluo-4AM dye based fluorescence assay | Homo sapiens | 26 | ALA4706753 | cell-based format | Scientific Literature | |
| 2. | ALA4715192 | F | Antagonist activity in CXCR1 (unknown origin) expressed in human HEK293 cells co-expressing Galpha16 assessed as reduction in calcium immobilization pretreated with Fluo-4AM for 45 mins followed by compound addition and measured after 10 mins by Fluo-4AM dye based fluorescence assay | Homo sapiens | 25 | ALA4706753 | cell-based format | Scientific Literature | |
| 3. | ALA4715193 | B | Selectivity index, ratio of IC50 for CXCR1 (unknown origin) expressed in human HEK293 cells to IC50 for CXCR2 (unknown origin) expressed in human HEK293 cells | Homo sapiens | 23 | ALA4706753 | cell-based format | Scientific Literature |
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