# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4714156 | B | Displacement of [3H]-gabapentin from human Cav alpha2delta1 expressed in CHO-K1 cell membranes incubated for 60 mins by scintillation counting method | Homo sapiens | 39 | cell membrane format | Scientific Literature | ||
2. | ALA4714157 | B | Displacement of [3H]-gabapentin from human Cav alpha2delta2 expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting method | Homo sapiens | 9 | cell membrane format | Scientific Literature | ||
3. | ALA4714158 | B | Displacement of [3H]-nisoxetine from human NET expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting method | Homo sapiens | 39 | cell membrane format | Scientific Literature | ||
4. | ALA4714159 | B | Inhibition of human NET expressed in HEK293 cells assessed as reduction in ASP+ uptake incubated for 20 mins before ASP+ addition and measured after 90 mins by scintillation counting method | Homo sapiens | 39 | cell-based format | Scientific Literature | ||
5. | ALA4714161 | A | Intrinsic clearance in human liver microsomes | Homo sapiens | 3 | microsome format | Scientific Literature | ||
6. | ALA4714162 | A | Intrinsic clearance in rat liver microsomes | Rattus norvegicus | 3 | microsome format | Scientific Literature | ||
7. | ALA4714163 | A | Inhibition of human CYP1A2 at 1 uM relative to control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
8. | ALA4714164 | A | Inhibition of human CYP2C9 at 1 uM relative to control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
9. | ALA4714165 | A | Inhibition of human CYP2C19 at 1 uM relative to control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
10. | ALA4714166 | A | Inhibition of human CYP2D6 at 1 uM relative to control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
11. | ALA4714167 | A | Inhibition of human CYP3A4 at 1 uM relative to control | Homo sapiens | 3 | single protein format | Scientific Literature | ||
12. | ALA4714168 | B | Inhibition of human ERG | Homo sapiens | 3 | single protein format | Scientific Literature |