| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4709751 | Binding | Inhibition of recombinant full length His-tagged human CDK9/cyclin T1 expressed in baculovirus expression system using biotinylated peptide biotin-Ttds-YISPLKSPYKISEG as substrate preincubated for 15 mins followed by ATP and substrate addition and measured after 25 mins by TR-FRET assay | Homo sapiens | 6 | ALA4706546 | assay format | Scientific Literature | |
| 2. | ALA4709752 | Binding | Inhibition of recombinant GST-tagged human CDK2/GST-tagged cyclin E expressed in sf9 cells using biotinylated peptide biotin-Ttds-YISPLKSPYKISEG as substrate preincubated for 15 mins followed by ATP and substrate addition and measured after 25 mins by TR-FRET assay | Homo sapiens | 5 | ALA4706546 | cell-based format | Scientific Literature | |
| 3. | ALA4709754 | Binding | Selectivity ratio of IC50 for GST-tagged human CDK2/GST-tagged cyclin E expressed in sf9 cells to IC50 for recombinant full length His-tagged human CDK9/cyclin T1 expressed in baculovirus expression system | Homo sapiens | 5 | ALA4706546 | cell-based format | Scientific Literature |
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