| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4709237 | B | Binding affinity to ERRgamma (unknown origin) by TR-FRET assay | Homo sapiens | 41 | single protein format | Scientific Literature | ||
| 2. | ALA4709238 | B | Inverse agonist activity at ERRgamma (unknown origin) assessed as receptor mediated luciferase activity at 10 uM by luciferase reporter gene assay relative to control | Homo sapiens | 29 | single protein format | Scientific Literature | ||
| 3. | ALA4709239 | B | Binding affinity to ERRalpha (unknown origin) by TR-FRET assay | Homo sapiens | 23 | single protein format | Scientific Literature | ||
| 4. | ALA4709240 | B | Binding affinity to ERRbeta (unknown origin) by TR-FRET assay | Homo sapiens | 23 | single protein format | Scientific Literature | ||
| 5. | ALA4709241 | B | Binding affinity to ERalpha (unknown origin) by TR-FRET assay | Homo sapiens | 23 | single protein format | Scientific Literature | ||
| 6. | ALA4709242 | B | Selectivity index, ratio of IC50 for ERRalpha (unknown origin) to IC50 for ERRgamma (unknown origin) | Homo sapiens | 8 | assay format | Scientific Literature | ||
| 7. | ALA4709243 | B | Selectivity index, ratio of IC50 for ERRbeta (unknown origin) to IC50 for ERRgamma (unknown origin) | Homo sapiens | 8 | assay format | Scientific Literature | ||
| 8. | ALA4709244 | B | Selectivity index, ratio of IC50 for ERalpha (unknown origin) to IC50 for ERRgamma (unknown origin) | Homo sapiens | 8 | assay format | Scientific Literature | ||
| 9. | ALA4709245 | A | Inhibition of CYP1A2 (unknown origin) in liver microsomes at 10 uM incubated for 15 mins relative to control | Homo sapiens | 10 | microsome format | Scientific Literature | ||
| 10. | ALA4709246 | A | Inhibition of CYP2C9 (unknown origin) in liver microsomes at 10 uM incubated for 15 mins relative to control | Homo sapiens | 10 | microsome format | Scientific Literature | ||
| 11. | ALA4709247 | A | Inhibition of CYP2C19 (unknown origin) in liver microsomes at 10 uM incubated for 15 mins relative to control | Homo sapiens | 10 | microsome format | Scientific Literature | ||
| 12. | ALA4709248 | A | Inhibition of CYP2D6 (unknown origin) in liver microsomes at 10 uM incubated for 15 mins relative to control | Homo sapiens | 10 | microsome format | Scientific Literature | ||
| 13. | ALA4709249 | A | Inhibition of CYP3A4 (unknown origin) in liver microsomes at 10 uM incubated for 15 mins relative to control | Homo sapiens | 10 | microsome format | Scientific Literature | ||
| 14. | ALA4709250 | A | Metabolic stability in human liver microsomes assessed as parent compound remaining | Homo sapiens | 9 | microsome format | Scientific Literature | ||
| 15. | ALA4709251 | A | Metabolic stability in dog liver microsomes assessed as parent compound remaining | Canis lupus familiaris | 9 | microsome format | Scientific Literature | ||
| 16. | ALA4709252 | A | Metabolic stability in rat liver microsomes assessed as parent compound remaining | Rattus norvegicus | 9 | microsome format | Scientific Literature | ||
| 17. | ALA4709253 | A | Metabolic stability in mouse liver microsomes assessed as parent compound remaining | Mus musculus | 9 | microsome format | Scientific Literature | ||
| 18. | ALA4709254 | A | Permeability of compound incubated for 5 hrs by PAMPA assay | 9 | assay format | Scientific Literature | |||
| 19. | ALA4709255 | B | Inhibition of human ERG by fluorescence polarization assay | Homo sapiens | 10 | single protein format | Scientific Literature | ||
| 20. | ALA4709256 | A | AUC in rat at 1 mg/kg, iv | Rattus norvegicus | 3 | organism-based format | Scientific Literature |
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