# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4768235 | Binding | Displacement of [3H]-(+)-pnetazocin from sigma1 receptor in guinea pig brain membrane incubated for 150 mins by liquid scintillation counting method | Cavia porcellus | 23 | ALA4765270 | cell membrane format | Scientific Literature | |
2. | ALA4768236 | Binding | Displacement of [3H]-diprenorphin from human mu opioid receptor expressed in CHO cell membrane incubated for 150 mins by liquid scintillation counting method | Homo sapiens | 23 | ALA4765270 | cell membrane format | Scientific Literature | |
3. | ALA4768237 | Binding | Inhibition of sigma 2 receptor (unknown origin) at 1 uM relative to control | Homo sapiens | 2 | ALA4765270 | assay format | Scientific Literature | |
4. | ALA4768238 | Binding | Inhibition of histamine H3 receptor (unknown origin) at 1 uM relative to control | Homo sapiens | 2 | ALA4765270 | single protein format | Scientific Literature | |
5. | ALA4768239 | Binding | Inhibition of 5HT1A receptor (unknown origin) at 1 uM relative to control | Homo sapiens | 2 | ALA4765270 | single protein format | Scientific Literature | |
6. | ALA4768240 | Binding | Inhibition of 5HT2A receptor (unknown origin) at 1 uM relative to control | Homo sapiens | 2 | ALA4765270 | single protein format | Scientific Literature | |
7. | ALA4768241 | Binding | Inhibition of 5-HT transporter (unknown origin) at 1 uM relative to control | Homo sapiens | 2 | ALA4765270 | single protein format | Scientific Literature | |
8. | ALA4768242 | Binding | Inhibition of noradrenaline transporter (unknown origin) at 1 uM relative to control | Homo sapiens | 2 | ALA4765270 | single protein format | Scientific Literature | |
9. | ALA4768243 | Binding | Inhibition of CB1 receptor (unknown origin) at 1 uM relative to control | Homo sapiens | 2 | ALA4765270 | single protein format | Scientific Literature | |
10. | ALA4768244 | Binding | Inhibition of CB2 receptor (unknown origin) at 1 uM relative to control | Homo sapiens | 2 | ALA4765270 | single protein format | Scientific Literature | |
11. | ALA4768245 | Binding | Inhibition of adrenergic alpha2 receptor (unknown origin) at 1 uM relative to control | Homo sapiens | 2 | ALA4765270 | assay format | Scientific Literature | |
12. | ALA4768246 | Binding | Inhibition of adrenergic alpha1 receptor (unknown origin) at 1 uM relative to control | Homo sapiens | 2 | ALA4765270 | assay format | Scientific Literature | |
13. | ALA4768247 | Binding | Inhibition of NMDA receptor (unknown origin) at 1 uM relative to control | Homo sapiens | 2 | ALA4765270 | assay format | Scientific Literature | |
14. | ALA4768248 | Toxicity | Toxicity in sc dosed ICR mouse assessed as mortality after 24 hrs | Mus musculus | 3 | ALA4765270 | organism-based format | Scientific Literature | |
15. | ALA4768249 | Functional | Antiallodynic activity against formalin-induced nociceptive behavior in ICR mouse assessed as licking/biting time at 50 mg/kg, sc pre-treated for 30 mins followed by formalin-stimulation and measured up to 5 mins | Mus musculus | 3 | ALA4765270 | organism-based format | Scientific Literature | |
16. | ALA4768250 | Functional | Antiallodynic activity against formalin-induced nociceptive behavior in ICR mouse assessed as licking/biting time at 50 mg/kg, sc pre-treated for 30 mins followed by formalin-stimulation and measured up to 15 to 30 mins | Mus musculus | 3 | ALA4765270 | organism-based format | Scientific Literature |