| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4701442 | B | Inhibition of CDK9 (unknown origin) using Ulight-labeled substrate by TR-FRET LANCE method | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 2. | ALA4701443 | B | Inhibition of CDK4 (unknown origin) using Ulight-labeled substrate by TR-FRET LANCE method | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 3. | ALA4701444 | B | Inhibition of CDK6 (unknown origin) using Ulight-labeled substrate by TR-FRET LANCE method | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 4. | ALA4701445 | B | Inhibition of CDK1 (unknown origin) using Ulight-labeled substrate by TR-FRET LANCE method | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 5. | ALA4701446 | B | Inhibition of CDK2 (unknown origin) using Ulight-labeled substrate by TR-FRET LANCE method | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 6. | ALA4701447 | B | Inhibition of CDK7 (unknown origin) using Ulight-labeled substrate by TR-FRET LANCE method | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 7. | ALA4701448 | B | Inhibition of CDK8 (unknown origin) by TR-FRET assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 8. | ALA4701449 | B | Selectivity ratio of IC50 for CDK1 (unknown origin) to CDK9 (unknown origin) | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 9. | ALA4701450 | B | Selectivity ratio of IC50 for CDK2 (unknown origin) to CDK9 (unknown origin) | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 10. | ALA4701451 | B | Selectivity ratio of IC50 for CDK7 (unknown origin) to CDK9 (unknown origin) | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 11. | ALA4701452 | B | Selectivity ratio of IC50 for CDK8 (unknown origin) to CDK9 (unknown origin) | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 12. | ALA4701453 | B | Selectivity ratio of IC50 for CDK4 (unknown origin) to CDK9 (unknown origin) | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 13. | ALA4701454 | B | Selectivity ratio of IC50 for CDK6 (unknown origin) to CDK9 (unknown origin) | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 14. | ALA4701456 | F | Antiproliferative activity against human NCI-H929 cells assessed as reduction in cell viability incubated for 24 hrs by Cell-Titer Glo assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 15. | ALA4701457 | F | Antiproliferative activity against human MV4-11 cells assessed as reduction in cell viability incubated for 24 hrs by Cell-Titer Glo assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 16. | ALA4701458 | A | Plasma clearance in Sprague-Dawley rat at 1 mg/kg, iv measured after 24 hrs by reverse phase HPLC analysis | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 17. | ALA4836671 | B | Inhibition of CDK9 (unknown origin) using Ulight-labeled substrate measured after 1.5 hrs by TR-FRET LANCE method | Homo sapiens | 24 | single protein format | Scientific Literature | ||
| 18. | ALA4836672 | F | Antiproliferative activity against human NCI-H929 cells assessed as reduction in cell viability incubated for 24 hrs by Cell-Titer Glo assay | Homo sapiens | 24 | cell-based format | Scientific Literature | ||
| 19. | ALA4836673 | B | Inhibition of CDK9 in human A-431 cells assessed as reduction in RNA polymerase2 phosphorylation at C-terminal ser2 residue incubated for 4 hrs by In-cell Western analysis | Homo sapiens | 23 | cell-based format | Scientific Literature | ||
| 20. | ALA4836674 | A | Half life in rat at 1 mg/kg, iv | Rattus norvegicus | 14 | organism-based format | Scientific Literature |
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