| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4772814 | B | Inhibition of PI3Kalpha (unknown origin) using PIP2 as substrate measured after 1 hr in presence of ATP by ADP-Glo reagent based assay | Homo sapiens | 15 | ALA4765397 | single protein format | Scientific Literature | |
| 2. | ALA4772815 | B | Inhibition of mTOR (unknown origin) using ULight-4E-BP1 as substrate measured after 45 mins in presence of ATP by LANCE Ultra assay | Homo sapiens | 13 | ALA4765397 | single protein format | Scientific Literature | |
| 3. | ALA4772816 | B | Inhibition of PI3Kbeta (unknown origin) using PIP2 as substrate measured after 1 hr in presence of ATP by ADP-Glo reagent based assay | Homo sapiens | 6 | ALA4765397 | single protein format | Scientific Literature | |
| 4. | ALA4772817 | B | Inhibition of PI3Kgamma (unknown origin) using PIP2 as substrate measured after 1 hr in presence of ATP by ADP-Glo reagent based assay | Homo sapiens | 6 | ALA4765397 | single protein format | Scientific Literature | |
| 5. | ALA4772818 | B | Inhibition of PI3Kdelta (unknown origin) using PIP2 as substrate measured after 1 hr in presence of ATP by ADP-Glo reagent based assay | Homo sapiens | 6 | ALA4765397 | single protein format | Scientific Literature | |
| 6. | ALA4772819 | F | Antiproliferative activity against human MDA-MB-231 cells assessed as reduction in cell viability after 48 hrs by MTT assay | Homo sapiens | 4 | ALA4765397 | cell-based format | Scientific Literature | |
| 7. | ALA4772820 | F | Antiproliferative activity against human HeLa cells assessed as reduction in cell viability after 48 hrs by MTT assay | Homo sapiens | 4 | ALA4765397 | cell-based format | Scientific Literature | |
| 8. | ALA4772821 | F | Antiproliferative activity against human CNE2 cells assessed as reduction in cell viability after 48 hrs by MTT assay | Homo sapiens | 4 | ALA4765397 | cell-based format | Scientific Literature | |
| 9. | ALA4772822 | F | Antiproliferative activity against human HCT116 cells assessed as reduction in cell viability after 48 hrs by MTT assay | Homo sapiens | 4 | ALA4765397 | cell-based format | Scientific Literature | |
| 10. | ALA4772823 | F | Antiproliferative activity against human HepG2 cells assessed as reduction in cell viability after 48 hrs by MTT assay | Homo sapiens | 4 | ALA4765397 | cell-based format | Scientific Literature | |
| 11. | ALA4772824 | F | Antiproliferative activity against human MCF-7 cells assessed as reduction in cell viability after 48 hrs by MTT assay | Homo sapiens | 4 | ALA4765397 | cell-based format | Scientific Literature | |
| 12. | ALA4772825 | B | Inhibition of PI3K/mTOR signaling in human HCT116 cells assessed as reduction in AKT phosphorylation at 10 uM measured by Western blot analysis | Homo sapiens | 2 | ALA4765397 | cell-based format | Scientific Literature | |
| 13. | ALA4772826 | B | Inhibition of PI3K/mTOR signaling in human HCT116 cells assessed as reduction in p7056K phosphorylation at 10 uM measured by Western blot analysis | Homo sapiens | 2 | ALA4765397 | cell-based format | Scientific Literature | |
| 14. | ALA4772827 | U | Metabolic stability in artificial gastrointestinal fluids | 4 | ALA4765397 | assay format | Scientific Literature | ||
| 15. | ALA4772828 | A | Metabolic stability in rat liver microsomes assessed as compound remaining measured after 45 mins | Rattus norvegicus | 4 | ALA4765397 | microsome format | Scientific Literature |
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