# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4673851 | B | Binding affinity to wild type SETD8 catalytic domain (unknown origin) (234 to 380 residues) expressed in Escherichia coli assessed as covalent adduct formation at 20 to 200 uM incubated for 3 hrs by LC-MSD-TOF analysis | Homo sapiens | 2 | assay format | Scientific Literature | ||
2. | ALA4673856 | B | Inhibition of recombinant SETD8 catalytic domain (unknown origin) (232 to 393 residues) expressed in Escherichia coli assessed as reduction in incorporation of [3H]-labeled methyl group into biotinylated H4 (1 to 24) peptide measured after 1 hr using [3H-SAM] by scintillation proximity assay | Homo sapiens | 3 | assay format | Scientific Literature |