| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4766422 | Binding | Inhibition of FLAG-tagged full-length HIF-PHD2 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotinyl-DLDLEMLAPYIPMDDDFQL as peptide substrates preincubated for 30 mins followed by substrate addition and measured after 2 hrs by LANCE assay | Homo sapiens | 25 | ALA4765235 | cell-based format | Scientific Literature | |
| 2. | ALA4766425 | Functional | In vivo inhibition of HIF-PHD2 in C57BL/6 mouse assessed as serum erythropoietin level at 15 mg/kg, iv measured after 4 hrs | Mus musculus | 14 | ALA4765235 | organism-based format | Scientific Literature | |
| 3. | ALA4766445 | ADME | Half life in dog at 1 mg/kg, po or 0.5 mg/kg, iv | Canis lupus familiaris | 5 | ALA4765235 | organism-based format | Scientific Literature |
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