| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4687834 | P | Kinetic solubility of the compound | 50 | ALA4680285 | small-molecule physicochemical format | Scientific Literature | ||
| 2. | ALA4687836 | A | Half life in mouse liver S9 fraction | Mus musculus | 13 | ALA4680285 | subcellular format | Scientific Literature | |
| 3. | ALA4687837 | B | Inhibition of PIM1 (unknown origin) by coupled kinetic assay | Homo sapiens | 52 | ALA4680285 | single protein format | Scientific Literature | |
| 4. | ALA4687838 | B | Binding affinity to recombinant PIM1 (unknown origin) assessed as thermal stability by measuring temperature shift at 10 uM by differential scanning fluorimetry | Homo sapiens | 43 | ALA4680285 | single protein format | Scientific Literature | |
| 5. | ALA4687839 | F | Antiproliferative activity against human MV4-11 cells | Homo sapiens | 50 | ALA4680285 | cell-based format | Scientific Literature | |
| 6. | ALA4687846 | B | Inhibition of human ERG | Homo sapiens | 5 | ALA4680285 | single protein format | Scientific Literature | |
| 7. | ALA4687849 | A | Efflux ratio of permeability in human Caco-2 cells | Homo sapiens | 9 | ALA4680285 | cell-based format | Scientific Literature | |
| 8. | ALA4687881 | A | Displacement of [3H]RX 821002 from rat brain adrenergic alpha 2 receptor at 10 uM incubated for 60 mins by radiometric scintillation analysis relative to control | Rattus norvegicus | 3 | ALA4680285 | tissue-based format | Scientific Literature | |
| 9. | ALA4687882 | A | Displacement of [125I]CCK-8s from recombinant human CCK1 at 10 uM incubated for 60 mins by radiometric scintillation analysis relative to control | Homo sapiens | 3 | ALA4680285 | single protein format | Scientific Literature | |
| 10. | ALA4687883 | A | Displacement of [3H]SCH 23390 from recombinant human dopamine D1 receptor at 10 uM incubated for 60 mins by radiometric scintillation analysis relative to control | Homo sapiens | 3 | ALA4680285 | single protein format | Scientific Literature | |
| 11. | ALA4687884 | A | Displacement of [3H]pyrilamine from recombinant human histamine H1 receptor at 10 uM incubated for 60 mins by radiometric scintillation analysis relative to control | Homo sapiens | 3 | ALA4680285 | single protein format | Scientific Literature | |
| 12. | ALA4687885 | A | Displacement of [3H]4-DAMP from recombinant human muscarinic M3 receptor at 10 uM incubated for 60 mins by radiometric scintillation analysis relative to control | Homo sapiens | 3 | ALA4680285 | single protein format | Scientific Literature | |
| 13. | ALA4687886 | A | Displacement of [125I]NKA from recombinant human NK2 receptor at 10 uM incubated for 60 mins by radiometric scintillation analysis relative to control | Homo sapiens | 3 | ALA4680285 | single protein format | Scientific Literature | |
| 14. | ALA4687887 | A | Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor at 10 uM incubated for 60 mins by radiometric scintillation analysis relative to control | Homo sapiens | 3 | ALA4680285 | single protein format | Scientific Literature | |
| 15. | ALA4687888 | A | Displacement of [3H]batrachotoxinin from rat Sodium channel site 2 at 10 uM incubated for 60 mins by radiometric scintillation analysis relative to control | Rattus norvegicus | 3 | ALA4680285 | assay format | Scientific Literature | |
| 16. | ALA4687889 | A | Displacement of [3H]nisoxetine from recombinant human norepinephrine transporter at 10 uM incubated for 120 mins by radiometric scintillation analysis relative to control | Homo sapiens | 3 | ALA4680285 | single protein format | Scientific Literature | |
| 17. | ALA4687890 | A | Displacement of [3H]BTCP from recombinant human dopamine transporter at 10 uM incubated for 120 mins by radiometric scintillation analysis relative to control | Homo sapiens | 3 | ALA4680285 | single protein format | Scientific Literature |
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