| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4689191 | B | Inhibition of human CDK5/p25 assessed as residual activity at 10 uM by ADP-Glo assay relative to control | Homo sapiens | 12 | protein complex format | Scientific Literature | ||
| 2. | ALA4689192 | B | Inhibition of human CDK9/CyclinT assessed as residual activity at 10 uM by ADP-Glo assay relative to control | Homo sapiens | 12 | protein complex format | Scientific Literature | ||
| 3. | ALA4689193 | B | Inhibition of human PIM1 assessed as residual activity at 10 uM by ADP-Glo assay relative to control | Homo sapiens | 12 | single protein format | Scientific Literature | ||
| 4. | ALA4689194 | B | Inhibition of mouse CLK1 assessed as residual activity at 10 uM by ADP-Glo assay relative to control | Mus musculus | 12 | single protein format | Scientific Literature | ||
| 5. | ALA4689195 | A | Inhibition of rat DYRK1A (1 to 499 residues) assessed as residual activity at 10 uM by ADP-Glo assay relative to control | Rattus norvegicus | 12 | single protein format | Scientific Literature | ||
| 6. | ALA4689196 | B | Inhibition of human HASPIN assessed as residual activity at 10 uM by ADP-Glo assay relative to control | Homo sapiens | 12 | single protein format | Scientific Literature | ||
| 7. | ALA4689197 | B | Inhibition of human GSK3beta assessed as residual activity at 10 uM by ADP-Glo assay relative to control | Homo sapiens | 12 | single protein format | Scientific Literature | ||
| 8. | ALA4689198 | B | Inhibition of human CK1epsilon assessed as residual activity at 10 uM by ADP-Glo assay relative to control | Homo sapiens | 12 | single protein format | Scientific Literature | ||
| 9. | ALA4689199 | B | Inhibition of recombinant human CLK1 (130 to end residues) using ERMRPRKRQGSVRRRV as substrate incubated for 40 mins in presence of [gamma33P-ATP] by scintillation counting analysis | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 10. | ALA4689200 | B | Inhibition of recombinant human CLK2 (138 to end residues) using YRRAAVPPSPSLSRHSSPHQS(p)EDEEE as substrate incubated for 40 mins in presence of [gamma33P-ATP] by scintillation counting analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA4689201 | B | Inhibition of recombinant human full length CLK3 using ERMRPRKRQGSVRRRV as substrate incubated for 40 mins in presence of [gamma33P-ATP] by scintillation counting analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA4689202 | B | Inhibition of recombinant human CLK4 (128 to end residues) using YRRAAVPPSPSLSRHSSPHQS(p)EDEEE as substrate incubated for 40 mins in presence of [gamma33P-ATP] by scintillation counting analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA4689203 | F | Cytotoxicity against human HuH-7 cells assessed as reduction in cell viability incubated for 48 hrs by Hoechst-33342 staining based cell counting method (Rvb > 25 microM) | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 14. | ALA4689204 | F | Cytotoxicity against human CaCo-2 cells assessed as reduction in cell viability incubated for 48 hrs by Hoechst-33342 staining based cell counting method (Rvb > 25 microM) | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 15. | ALA4689205 | F | Cytotoxicity against human MDA-MB-231 cells assessed as reduction in cell viability incubated for 48 hrs by Hoechst-33342 staining based cell counting method (Rvb > 25 microM) | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 16. | ALA4689206 | F | Cytotoxicity against human HCT-116 cells assessed as reduction in cell viability incubated for 48 hrs by Hoechst-33342 staining based cell counting method (Rvb > 25 microM) | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 17. | ALA4689207 | F | Cytotoxicity against human PC-3 cells assessed as reduction in cell viability incubated for 48 hrs by Hoechst-33342 staining based cell counting method (Rvb > 25 microM) | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 18. | ALA4689208 | F | Cytotoxicity against human NCI-H727 cells assessed as reduction in cell viability incubated for 48 hrs by Hoechst-33342 staining based cell counting method (Rvb > 25 microM) | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 19. | ALA4689209 | F | Cytotoxicity against human MCF7 cells assessed as reduction in cell viability incubated for 48 hrs by Hoechst-33342 staining based cell counting method (Rvb > 25 microM) | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 20. | ALA4689210 | A | Cytotoxicity against human Fibroblast cells assessed as reduction in cell viability incubated for 48 hrs by Hoechst-33342 staining based cell counting method (Rvb > 25 microM) | Homo sapiens | 10 | cell-based format | Scientific Literature |
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