| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4775829 | B | Inhibition of human GRK5 using porcine brain tubulin as substrate incubated for 3 to 5 mins by [gamma32P]ATP based radiometric assay | Homo sapiens | 31 | assay format | Scientific Literature | ||
| 2. | ALA4775830 | B | Inhibition of bovine GRK2 using porcine brain tubulin as substrate incubated for 3 to 5 mins by [gamma32P]ATP based radiometric assay | Bos taurus | 31 | assay format | Scientific Literature | ||
| 3. | ALA4775831 | B | Selectivity index, ratio of IC50 for bovine GRK2 to IC50 for human GRK5 using porcine brain tubulin as substrate by [gamma-32P]-ATP assay | 29 | assay format | Scientific Literature | |||
| 4. | ALA4775834 | B | Covalent binding affinity to GRK5 (unknown origin) assessed as covalent adduct formation at 1 mM measured at 30 mins by LC/MS analysis | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 5. | ALA4775836 | B | Covalent inhibition of GRK5 (unknown origin) using porcine brain tubulin as substrate by [gamma32P]ATP based radiometric assay | Homo sapiens | 3 | assay format | Scientific Literature | ||
| 6. | ALA4775837 | B | Inhibition of human GRK5 C474S mutant using porcine brain tubulin as substrate incubated for 3 to 5 mins by [gamma32P]ATP based radiometric assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 7. | ALA4775838 | B | Selectivity index, ratio of IC50 for human GRK5 C474S mutant to IC50 for human GRK5 using porcine brain tubulin as substrate by [gamma32P]ATP based radiometric assay | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 8. | ALA4775842 | B | Inhibition of human GRK5 using porcine brain tubulin as substrate incubated for 3 to 5 mins at 1 uM by [gamma32P]ATP based radiometric assay relative to control | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 9. | ALA4775843 | B | Inhibition of GRK3 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA4775844 | B | Inhibition of GRK6 (unknown origin) at 1 uM relative to control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 11. | ALA4775845 | B | Inhibition of PKA (unknown origin) incubated for 30 mins using REBtide substrate by ADP-Glo assay | Homo sapiens | 31 | assay format | Scientific Literature |
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