| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4667069 | B | Inhibition of tracer 236 binding to recombinant human GST-tagged full length CAMKK2 expressed in baculovirus expression system at 10 uM incubated for 60 mins by Lanthascreen assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 2. | ALA4667070 | B | Inhibition of tracer 236 binding to recombinant human GST-tagged full length CAMKK1 expressed in Escherichia coli expression system at 10 uM incubated for 60 mins by Lanthascreen assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 3. | ALA4667071 | B | Inhibition of recombinant human His-tagged full length BRK expressed in baculovirus expression system using Tyr 01 as substrate at 10 uM incubated for 60 mins by Z'-Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 4. | ALA4667072 | B | Inhibition of recombinant human GST-tagged full length BrSK1 expressed in baculovirus expression system using Ser/Thr 21 as substrate at 10 uM incubated for 60 mins by Z'-Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 5. | ALA4667073 | B | Inhibition of recombinant human His-tagged full length BMX expressed in baculovirus expression system using Tyr 01 as substrate at 10 uM incubated for 60 mins by Z'-Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 6. | ALA4667074 | B | Inhibition of recombinant human His-tagged full length BLK expressed in baculovirus expression system using Tyr 01 as substrate at 10 uM incubated for 60 mins by Z'-Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 7. | ALA4667075 | B | Inhibition of recombinant human His-tagged full length BTK expressed in baculovirus expression system using Tyr 01 as substrate at 10 uM incubated for 60 mins by Z'-Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 8. | ALA4667076 | B | Inhibition of recombinant human GST-tagged full length BRAF expressed in baculovirus expression system using Ser/Thr 03 as substrate at 10 uM incubated for 60 mins by Z'-Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 9. | ALA4667077 | B | Inhibition of tracer 178 binding to recombinant human N-terminal GST-tagged full length BMPR1A expressed in insect expression system at 10 uM incubated for 60 mins by Lanthascreen assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 10. | ALA4667078 | B | Inhibition of recombinant human GST-tagged full length AXL expressed in insect expression system using Tyr 06 as substrate at 10 uM incubated for 60 mins by Z'-Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 11. | ALA4667079 | B | Inhibition of recombinant human His-tagged full length Aurora B expressed in baculovirus expression system using Ser/Thr 01 as substrate at 10 uM incubated for 60 mins by Z'-Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 12. | ALA4667080 | B | Inhibition of recombinant human N-terminal GST-tagged full length JNK3 expressed in baculovirus expression system using Ser/Thr 04 as substrate at 10 uM incubated for 60 mins by Z'-lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 13. | ALA4667081 | B | Inhibition of recombinant human His-tagged KDR (789 to 1356 residues) expressed in baculovirus expression system using Tyr 01 as substrate at 10 uM incubated for 60 mins by Z'-lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA4667082 | B | Inhibition of recombinant human His-tagged full length Aurora A expressed in baculovirus expression system using Ser/Thr 01 as substrate at 10 uM incubated for 60 mins by Z'-Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA4667083 | B | Inhibition of recombinant human His-tagged full length Abl expressed in baculovirus expression system using Tyr 02 as substrate at 10 uM incubated for 60 mins by Z'-Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 16. | ALA4667084 | B | Inhibition of tracer 236 binding to recombinant human GST-tagged full length ASK1 expressed in baculovirus expression system at 10 uM incubated for 60 mins by Lanthascreen assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 17. | ALA4667085 | B | Inhibition of recombinant human GST-tagged ACVR1B (150 to 505 residues) expressed in baculovirus expression system using Ser/Thr 16 as substrate at 10 uM incubated for 60 mins by Z'-Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 18. | ALA4667086 | F | Inhibition of necroptosis in mouse L929 cells assessed as reduction in TNFalpha/BV6/zVAD-fmk-induced cell death incubated for 18 hrs by Cell Titer Glo luminescent cell viability assay | Mus musculus | 1 | cell-based format | Scientific Literature | ||
| 19. | ALA4667087 | B | Inhibition of mouse RIPK1 incubated for 2 hrs by fluorescence polarization assay | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 20. | ALA4667088 | A | Half life in Sprague-Dawley rat at 0.5 mg/kg, iv or 2 mg/kg, po | Rattus norvegicus | 1 | organism-based format | Scientific Literature |
The page will load shortly, Thanks for your patience!