| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4725002 | Binding | Inhibition of human SGLT2 expressed in COS7 cells assessed as reduction in [14C]-AMG uptake | Homo sapiens | 24 | ALA4715919 | cell-based format | Scientific Literature | |
| 2. | ALA4725003 | Binding | Inhibition of human SGLT1 expressed in COS7 cells assessed as reduction in [14C]-AMG uptake | Homo sapiens | 24 | ALA4715919 | cell-based format | Scientific Literature | |
| 3. | ALA4725004 | Binding | Selectivity ratio IC50 for human SGLT1 expressed in COS7 cells to IC50 for human SGLT2 expressed in COS7 cells | Homo sapiens | 22 | ALA4715919 | cell-based format | Scientific Literature | |
| 4. | ALA4725006 | ADME | Intrinsic clearance in human liver microsomes at 30 uM up to 60 mins by LC-MS/MS analysis | Homo sapiens | 6 | ALA4715919 | microsome format | Scientific Literature |
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