#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA4670919	A	Ratio of apparent permeability across basolateral to apical over apical to basolateral side in human Caco2 cells at 5 uM after 2 hrs by transwell assay	Homo sapiens	8	ALA4665812	cell-based format	Scientific Literature
2.	ALA4670920	A	Apparent permeability across apical side to basolateral side in human Caco-2 cells at 5 uM after 2 hrs by transwell assay	Homo sapiens	8	ALA4665812	cell-based format	Scientific Literature
3.	ALA4670921	A	Intrinsic clearance in mouse liver microsomes at 3 uM measured up to 60 mins by LC-MS analysis	Mus musculus	5	ALA4665812	microsome format	Scientific Literature
4.	ALA4670922	A	Intrinsic clearance in human liver microsomes at 3 uM measured up to 50 mins by LC-MS analysis	Homo sapiens	5	ALA4665812	microsome format	Scientific Literature
5.	ALA4670923	A	Stability of compound in mouse plasma assessed as parent compound remaining at 5 uM measured for 1 hr by LC-MS analysis	Mus musculus	8	ALA4665812	cell-free format	Scientific Literature
6.	ALA4670924	A	Stability of compound in human plasma assessed as parent compound remaining at 5 uM measured for 1 hr by LC-MS analysis	Homo sapiens	8	ALA4665812	cell-free format	Scientific Literature
7.	ALA4670925	P	Kinetic solubility of compound in HEPES buffer a pH 7.4 at 500 uM after 90 mins		8	ALA4665812	small-molecule physicochemical format	Scientific Literature
8.	ALA4670926	P	Solubility of compound in aqueous buffer at pH 7.4 after 120 mins by turbidometric assay		8	ALA4665812	small-molecule physicochemical format	Scientific Literature
9.	ALA4670927	B	Inhibiton of EGFR L858R/T790M mutant (unknown origin) expressed in human NCI-H1975 cells assessed as reduction in EGFR induced cell viability after 96 hrs by CellTiter-Glo assay	Homo sapiens	8	ALA4665812	cell-based format	Scientific Literature
10.	ALA4670928	B	Inhibiton of EGFR (unknown origin) expressed in human A431 cells assessed as reduction in EGFR induced cell viability after 96 hrs by CellTiter-Glo assay	Homo sapiens	8	ALA4665812	cell-based format	Scientific Literature
11.	ALA4670929	B	Inhibition of human N-terminal GST-tagged EGFR L858R/T790M mutant (669 to 1210 residues) expressed in baculovirus infected Sf9 insect cells using TK as substrate preincubated for 30 mins followed by substrate addition and measured after 20 mins by HTRF assay	Homo sapiens	8	ALA4665812	cell-based format	Scientific Literature
12.	ALA4670930	B	Inhibition of human N-terminal GST-tagged EGFR L858R mutant (669 to 1210 residues) expressed in baculovirus infected Sf9 insect cells using TK as substrate preincubated for 30 mins followed by substrate addition and measured after 15 mins by HTRF assay	Homo sapiens	8	ALA4665812	cell-based format	Scientific Literature
13.	ALA4670931	B	Inhibition of human N-terminal GST-tagged EGFR (669 to 1210 residues) expressed in baculovirus infected Sf9 insect cells using TK as substrate preincubated for 30 mins followed by substrate addition and measured after 25 mins by HTRF assay	Homo sapiens	8	ALA4665812	cell-based format	Scientific Literature
14.	ALA4670932	B	Potency index, ratio of neratinib Kinact to test compound Kinact for inhibition of C-terminal His6-tagged HER2-A775_G776insYVMA mutant (703 to 1029 residues) (unknown origin) expressed in Sf9 insect cells	Homo sapiens	4	ALA4665812	cell-based format	Scientific Literature
15.	ALA4670933	B	Potency index, ratio of afatinib Kinact to test compound Kinact for inhibition of C-terminal His6-tagged HER2-A775_G776insYVMA mutant (703 to 1029 residues) (unknown origin) expressed in Sf9 insect cells	Homo sapiens	4	ALA4665812	cell-based format	Scientific Literature
16.	ALA4670934	B	Inhibition of C-terminal His6-tagged HER2-A775_G776insYVMA mutant (703 to 1029 residues) (unknown origin) expressed in Sf9 insect cells assessed as ratio of Kinact to Ki using TK as substrate measured up to 2 to 40 mins by fluorescence assay	Homo sapiens	6	ALA4665812	cell-based format	Scientific Literature
17.	ALA4670935	B	Inhibition of C-terminal His6-tagged HER2-A775_G776insYVMA mutant (703 to 1029 residues) (unknown origin) expressed in Sf9 insect cells assessed as Kinact using TK as substrate measured up to 2 to 40 mins by fluorescence assay	Homo sapiens	6	ALA4665812	cell-based format	Scientific Literature
18.	ALA4670936	B	Inhibition of C-terminal His6-tagged HER2-A775_G776insYVMA mutant (703 to 1029 residues) (unknown origin) expressed in Sf9 insect cells using TK as substrate measured up to 2 to 40 mins by fluorescence assay	Homo sapiens	6	ALA4665812	cell-based format	Scientific Literature
19.	ALA4670939	B	Inhibition of S6 phosphorylation at T202/204 residues in human H1781 cells after 1 hrs by Western blot analysis	Homo sapiens	2	ALA4665812	cell-based format	Scientific Literature
20.	ALA4670940	B	Inhibition of MAPK phosphorylation at T202/204 residues in human H1781 cells after 1 hrs by Western blot analysis	Homo sapiens	2	ALA4665812	cell-based format	Scientific Literature