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# Aladdin ID Assay Type Description Organism Compounds Reference BAO Format Source 1. ALA4708712 B Binding affinity to androgen receptor (unknown origin) 10 umol/L by radioligand binding assay Homo sapiens 2 single protein format Scientific Literature 2. ALA4708713 B Binding affinity to AT2 receptor (unknown origin) 10 umol/L by radioligand binding assay Homo sapiens 2 single protein format Scientific Literature 3. ALA4708714 B Binding affinity to AT1 receptor (unknown origin) 10 umol/L by radioligand binding assay Homo sapiens 2 single protein format Scientific Literature 4. ALA4708715 B Binding affinity to beta2 adrenoreceptor (unknown origin) 10 umol/L by radioligand binding assay Homo sapiens 2 single protein format Scientific Literature 5. ALA4708716 B Binding affinity to beta1 adrenoreceptor (unknown origin) 10 umol/L by radioligand binding assay Homo sapiens 2 single protein format Scientific Literature 6. ALA4708717 B Binding affinity to alpha2C adrenoreceptor (unknown origin) 10 umol/L by radioligand binding assay Homo sapiens 2 single protein format Scientific Literature 7. ALA4708718 B Binding affinity to alpha2A adrenoreceptor (unknown origin) 10 umol/L by radioligand binding assay Homo sapiens 2 single protein format Scientific Literature 8. ALA4708719 B Binding affinity to alpha1B adrenoreceptor (unknown origin) 10 umol/L by radioligand binding assay Homo sapiens 2 single protein format Scientific Literature 9. ALA4708720 B Binding affinity to adenosine transporter (unknown origin) at 10 umol/L by radioligand binding assay Homo sapiens 2 assay format Scientific Literature 10. ALA4708721 B Binding affinity to alpha1A adrenoreceptor (unknown origin) 10 umol/L by radioligand binding assay Homo sapiens 2 single protein format Scientific Literature 11. ALA4708722 B Binding affinity to A3 receptor (unknown origin) 10 umol/L by radioligand binding assay Homo sapiens 2 single protein format Scientific Literature 12. ALA4708723 B Binding affinity to A1 receptor (unknown origin) at 10 umol/L by radioligand binding assay Homo sapiens 2 single protein format Scientific Literature 13. ALA4708724 B Binding affinity to A2a receptor (unknown origin) at 10 umol/L by radioligand binding assay Homo sapiens 2 single protein format Scientific Literature 14. ALA4708725 B Binding affinity to alpha2B adrenoreceptor (unknown origin) 10 umol/L by radioligand binding assay Homo sapiens 2 single protein format Scientific Literature 15. ALA4708727 A Prodrug conversion in monkey liver microsomes assessed as formation of (1S,2S,3S,5R,6S)-2-amino-3-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylicacid at 3 umol/L after 15 mins by LC-MS/MS analysis Macaca mulatta 13 microsome format Scientific Literature 16. ALA4708728 A Prodrug conversion in human liver microsomes assessed as formation of (1S,2S,3S,5R,6S)-2-amino-3-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylicacid at 3 umol/L after 15 mins by LC-MS/MS analysis Homo sapiens 13 microsome format Scientific Literature 17. ALA4708729 P Stability of compound in HCL at pH 1.2 assessed as remaining parent compound at 50 ug/ml after 1 hr by HPLC analysis 13 small-molecule physicochemical format Scientific Literature 18. ALA4708730 P Stability of compound in PBS at pH 6.5 assessed as remaining parent compound at 50 ug/ml after 1 hr by HPLC analysis 13 small-molecule physicochemical format Scientific Literature 19. ALA4708731 P Lipophilicity, logD of compound in n-octanol and phosphate buffered saline at 2 mg after 1.5 hrs by HPLC based shake flask method 13 small-molecule physicochemical format Scientific Literature 20. ALA4708732 F Agonist activity at human mGlu2 receptor expressed in CHO cell membranes by GTPgammaS binding assay Homo sapiens 2 cell membrane format Scientific Literature