| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4723883 | B | Inhibition of PIM1 (unknown origin) using Bad peptide NH2-AGAGRSRHSSYPAGT-OH as substrate measured after 10 mins in presence of ATP by luciferase-luciferin based Kinase-Glo luminescence assay | Homo sapiens | 14 | single protein format | Scientific Literature | ||
| 2. | ALA4723884 | B | Inhibition of PIM2 (unknown origin) using Bad peptide NH2-AGAGRSRHSSYPAGT-OH as substrate measured after 10 mins in presence of ATP by luciferase-luciferin based Kinase-Glo luminescence assay | Homo sapiens | 14 | single protein format | Scientific Literature | ||
| 3. | ALA4723885 | B | Inhibition of PIM3 (unknown origin) using Bad peptide NH2-AGAGRSRHSSYPAGT-OH as substrate measured after 10 mins in presence of ATP by luciferase-luciferin based Kinase-Glo luminescence assay | Homo sapiens | 14 | single protein format | Scientific Literature | ||
| 4. | ALA4723886 | F | Antiproliferative activity against human KMS-11 cells expressing firefly luciferase assessed as reduction in cell viability incubated for 72 hrs by cell titer-glo assay | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
| 5. | ALA4723887 | P | Lipophilicity, log D of the compound at pH 7.4 | 14 | small-molecule physicochemical format | Scientific Literature | |||
| 6. | ALA4723888 | A | Intrinsic clearance in rat liver microsomes at 1 uM incubated for 30 mins in presence of NADPH by LC-MS/MS analysis | Rattus norvegicus | 14 | microsome format | Scientific Literature | ||
| 7. | ALA4723889 | A | Intrinsic clearance in human liver microsomes at 1 uM incubated for 30 mins in presence of NADPH by LC-MS/MS analysis | Homo sapiens | 14 | microsome format | Scientific Literature | ||
| 8. | ALA4723890 | A | Hepatic extraction ratio in rat liver microsomes at 1 uM incubated for 30 mins in presence of NADPH by LC-MS/MS analysis | Rattus norvegicus | 14 | microsome format | Scientific Literature | ||
| 9. | ALA4723891 | A | Hepatic extraction ratio in human liver microsomes at 1 uM incubated for 30 mins in presence of NADPH by LC-MS/MS analysis | Homo sapiens | 14 | microsome format | Scientific Literature | ||
| 10. | ALA4723892 | A | Apparent permeability from apical to basolateral side in human Caco2 cells | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
| 11. | ALA4723893 | A | Efflux ratio of apparent permeability across basolateral to apical side over apical to basolateral side in human Caco2 cells | Homo sapiens | 14 | cell-based format | Scientific Literature |
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