| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4839006 | B | Inhibition of recombinant FAK (unknown origin) by radiometric kinase assay | Homo sapiens | 42 | single protein format | Scientific Literature | ||
| 2. | ALA4839008 | F | Antiproliferative activity against human HCT-116 cells assessed as growth inhibition measured after 72 hrs by CellTiter-Glo assay | Homo sapiens | 34 | cell-based format | Scientific Literature | ||
| 3. | ALA4839009 | F | Antiproliferative activity against human MDA-MB-231 cells assessed as growth inhibition measured after 72 hrs by CellTiter-Glo assay | Homo sapiens | 34 | cell-based format | Scientific Literature | ||
| 4. | ALA4839010 | F | Antiproliferative activity against human A375P cells assessed as growth inhibition measured after 72 hrs by CellTiter-Glo assay | Homo sapiens | 34 | cell-based format | Scientific Literature | ||
| 5. | ALA4839011 | A | Metabolic stability in human liver microsomes assessed as compound remaining at 1 uM measured after 1 hr | Homo sapiens | 21 | microsome format | Scientific Literature | ||
| 6. | ALA4839012 | B | Inhibition of FYK Y379 mutant phosphorylation in human HCT-116 cells by Western blot analysis | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 7. | ALA4839013 | B | Inhibition of FYK Y379 mutant phosphorylation in human MDA-MB-231 cells by Western blot analysis | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 8. | ALA4839014 | B | Inhibition of FYK Y379 mutant phosphorylation in human MDA-MB-231 cells by in-cell western blot assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 9. | ALA4839015 | A | Inhibition of CYP1A2 (unknown origin) at 10 uM relative to control | Homo sapiens | 10 | single protein format | Scientific Literature | ||
| 10. | ALA4839016 | A | Inhibition of CYP2C9 (unknown origin) at 10 uM relative to control | Homo sapiens | 10 | single protein format | Scientific Literature | ||
| 11. | ALA4839017 | A | Inhibition of CYP2C19 (unknown origin) at 10 uM relative to control | Homo sapiens | 10 | single protein format | Scientific Literature | ||
| 12. | ALA4839018 | A | Inhibition of CYP2D6 (unknown origin) at 10 uM relative to control | Homo sapiens | 10 | single protein format | Scientific Literature | ||
| 13. | ALA4839019 | A | Inhibition of CYP3A4 (unknown origin) at 10 uM relative to control | Homo sapiens | 10 | single protein format | Scientific Literature | ||
| 14. | ALA4839020 | B | Inhibition of human ERG by patch-clamp assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA4839021 | A | Oral bioavailability in mouse at 10 mg/kg | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 16. | ALA4839022 | A | Oral bioavailability in rat at 5 mg/kg | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 17. | ALA4839023 | B | Inhibition of FLT3 D835Y (unknown origin) | Homo sapiens | 15 | assay format | Scientific Literature | ||
| 18. | ALA4839024 | B | Inhibition of DDR1 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA4839025 | B | Inhibition of JAK3 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 20. | ALA4839026 | B | Inhibition of TYK2 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature |
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