# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4832445 | Binding | Displacement of [3H]-DPN from mouse kappa opioid receptor stably expressed in HEK293 cell membrane at 10 uM incubated for 1 hr by radioligand competition binding based assay | Mus musculus | 6 | ALA4831505 | cell membrane format | Scientific Literature | |
2. | ALA4832446 | Binding | Displacement of [3H]-DPN from mouse kappa opioid receptor stably expressed in HEK293 cell membrane assessed as inhibition constant incubated for 1 hr by radioligand competition binding based assay | Mus musculus | 2 | ALA4831505 | cell membrane format | Scientific Literature | |
3. | ALA4832447 | Functional | Agonist activity at mouse kappa opioid receptor stably expressed in HEK293 cell membrane assessed as inhibition of forskolin induced cAMP production by measuring maximum efficacy incubated for 30 mins by HTRF assay relative to control | Mus musculus | 2 | ALA4831505 | cell membrane format | Scientific Literature | |
4. | ALA4832448 | Functional | Agonist activity at mouse kappa opioid receptor stably expressed in HEK293 cell membrane assessed as inhibition of forskolin induced cAMP production incubated for 30 mins by HTRF assay | Mus musculus | 2 | ALA4831505 | cell membrane format | Scientific Literature |