# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4824985 | Binding | Inhibition of human PDHK2 co-complexed with porcine PDH using sodium pyruvate, coenzymeA and NAD as substrate preincubated with enzyme complex for 45 mins followed by ATP addition and then later incubated with substrate for 90 mins by absorption spectrophotometric assay | Homo sapiens | 16 | ALA4823293 | single protein format | Scientific Literature | |
2. | ALA4824986 | Binding | Inhibition of human PDHK4 co-complexed with porcine PDH using sodium pyruvate, coenzymeA and NAD as substrate preincubated with enzyme complex for 45 mins followed by ATP addition and then later incubated with substrate for 90 mins by absorption spectrophotometric assay | Homo sapiens | 16 | ALA4823293 | single protein format | Scientific Literature | |
3. | ALA4824989 | Binding | Inhibition of human PDHK1 co-complexed with porcine PDH using sodium pyruvate, coenzymeA and NAD as substrate preincubated with enzyme complex for 45 mins followed by ATP addition and then later incubated with substrate for 90 mins by absorption spectrophotometric assay | Homo sapiens | 1 | ALA4823293 | single protein format | Scientific Literature | |
4. | ALA4824990 | Binding | Inhibition of human PDHK3 co-complexed with porcine PDH using sodium pyruvate, coenzymeA and NAD as substrate preincubated with enzyme complex for 45 mins followed by ATP addition and then later incubated with substrate for 90 mins by absorption spectrophotometric assay | Homo sapiens | 1 | ALA4823293 | single protein format | Scientific Literature | |
5. | ALA4824992 | Binding | Inhibition of HSP90 (unknown origin) at 30 uM using labelled geldanamycin by fluorescence polarization assay | Homo sapiens | 1 | ALA4823293 | protein format | Scientific Literature | |
6. | ALA4824993 | Binding | Inhibition of human recombinant BCKDK at 500 uM incubated for 60 mins by ADP-Glo kinase assay | Homo sapiens | 1 | ALA4823293 | single protein format | Scientific Literature | |
7. | ALA4824994 | Binding | Inhibition of human partial length wild type mTOR (L1382 to W2549 residues) expressed in mammalian expression system at 10 uM by KINOMEscan analysis | Homo sapiens | 1 | ALA4823293 | assay format | Scientific Literature | |
8. | ALA4824995 | Binding | Inhibition of human partial length wild type MAST1 (S346 to V730 residues) expressed in mammalian expression system at 10 uM by KINOMEscan analysis | Homo sapiens | 1 | ALA4823293 | assay format | Scientific Literature |