# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4808118 | Functional | Antagonist activity at human MRGPRX4 expressed in HEK cells incubated in dark for 1 hr at 37 degree C and then incubated for 30 mins at room temperature in presence of 10 pM of bilirubin by HTRF assay | Homo sapiens | 309 | ALA4806969 | cell-based format | Patent Bioactivity Data | |
2. | ALA4808119 | Functional | Antagonist activity at human MRGPRX4 expressed in HEK cells incubated in dark for 1 hr at 37 degree C and then incubated for 30 mins at room temperature in presence of 10 uM of bilirubin by HTRF assay | Homo sapiens | 17 | ALA4806969 | cell-based format | Patent Bioactivity Data | |
3. | ALA4808120 | Functional | Antagonist activity at human MRGPRX4 expressed in HEK cells incubated in dark for 1 hr at 37 degree C and then incubated for 30 mins at room temperature in presence of 100 uM of conjugated bilirubin by HTRF assay | Homo sapiens | 17 | ALA4806969 | cell-based format | Patent Bioactivity Data | |
4. | ALA4808121 | Functional | Antagonist activity at human MRGPRX4 expressed in HEK cells incubated in dark for 1 hr at 37 degree C and then incubated for 30 mins at room temperature in presence of 20 uM of deoxycholic acid by HTRF assay | Homo sapiens | 17 | ALA4806969 | cell-based format | Patent Bioactivity Data | |
5. | ALA4808122 | Functional | Antagonist activity at human MRGPRX4 expressed in HEK cells incubated in dark for 1 hr at 37 degree C and then incubated for 30 mins at room temperature in presence of 50 uM of urobilin by HTRF assay | Homo sapiens | 17 | ALA4806969 | cell-based format | Patent Bioactivity Data | |
6. | ALA4808123 | Functional | Antagonist activity at human MRGPRX4 expressed in HEK cells incubated in dark for 1 hr at 37 degree C and then incubated for 30 mins at room temperature in presence of 50 uM of obeticholic acid by HTRF assay | Homo sapiens | 17 | ALA4806969 | cell-based format | Patent Bioactivity Data | |
7. | ALA4808127 | Functional | Antagonist activity at human MRGPRX4 expressed in HEK cells incubated in dark for 1 hr at 37 degree C and then incubated for 30 mins at room temperature in presence of 10 uM of BAR-502 by HTRF assay | Homo sapiens | 8 | ALA4806969 | cell-based format | Patent Bioactivity Data |