| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4839297 | Functional | Antagonist activity at human muscarinic M2 receptor expressed in CHO cells co-expressing Gqi5 assessed as inhibition of acetylcholine-induced calcium mobilization | Homo sapiens | 11 | ALA4837245 | cell-based format | Scientific Literature | |
| 2. | ALA4839302 | ADME | Efflux ratio of apparent permeability basolateral to apical over apical to basolateral side at human P-gp in MDCK-MDR1 cells | Canis lupus familiaris | 12 | ALA4837245 | cell-based format | Scientific Literature | |
| 3. | ALA4839303 | Functional | Antagonist activity at human muscarinic acetylcholine M4 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilization | Homo sapiens | 12 | ALA4837245 | cell-based format | Scientific Literature | |
| 4. | ALA4839304 | Binding | Antagonist activity at human muscarinic acetylcholine M4 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilization relative to control | Homo sapiens | 12 | ALA4837245 | cell-based format | Scientific Literature | |
| 5. | ALA4839336 | Binding | Selectivity index, ratio of IC50 for human muscarinic receptor M2 expressed in CHO cells to IC50 for human muscarinic receptor M4 expressed in CHO cells | Homo sapiens | 11 | ALA4837245 | cell-based format | Scientific Literature |
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