| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4840464 | B | Inhibition of N-terminal GST-tagged human TRKA (436 to 790 residues) expressed in baculovirus infected Sf21 cells using TK as substrate in presence of ATP measured after 30 mins by HTRF assay | Homo sapiens | 43 | ALA4840303 | cell-based format | Scientific Literature | |
| 2. | ALA4840465 | B | Inhibition of N-terminal GST-tagged human TRKB (456 to 822 residues) expressed in baculovirus infected Sf21 cells using TK as substrate in presence of ATP measured after 40 mins by HTRF assay | Homo sapiens | 7 | ALA4840303 | cell-based format | Scientific Literature | |
| 3. | ALA4840466 | B | Inhibition of N-terminal GST-tagged human TRKC (456 to 825 residues) expressed in Sf21 using TK as substrate in presence of ATP measured after 40 mins by HTRF assay | Homo sapiens | 7 | ALA4840303 | cell-based format | Scientific Literature | |
| 4. | ALA5053785 | B | Inhibition of TRKA F589L mutant (unknown origin) in presence of [gamma-33P]ATP by hotspot kinase assay | Homo sapiens | 2 | ALA5053493 | assay format | Scientific Literature | |
| 5. | ALA5053786 | B | Inhibition of TRKC G623R mutant (unknown origin) in presence of [gamma-33P]ATP by hotspot kinase assay | Homo sapiens | 2 | ALA5053493 | assay format | Scientific Literature | |
| 6. | ALA5053787 | B | Inhibition of TRKC G696A mutant (unknown origin) in presence of [gamma-33P]ATP by hotspot kinase assay | Homo sapiens | 2 | ALA5053493 | assay format | Scientific Literature | |
| 7. | ALA5053788 | B | Inhibition of TRKC L686M mutant (unknown origin) in presence of [gamma-33P]ATP by hotspot kinase assay | Homo sapiens | 2 | ALA5053493 | assay format | Scientific Literature | |
| 8. | ALA5053789 | B | Inhibition of TRKA G595R/A608D double mutant (unknown origin) bin presence of [gamma-33P]ATP by hotspot kinase assay | Homo sapiens | 2 | ALA5053493 | assay format | Scientific Literature | |
| 9. | ALA5053790 | B | Inhibition of TRKA GS95R/G667C double mutant (unknown origin) in presence of [gamma-33P]ATP by hotspot kinase assay | Homo sapiens | 2 | ALA5053493 | assay format | Scientific Literature | |
| 10. | ALA5053791 | B | Inhibition of TRKA G595R/L657M double mutant(unknown origin) in presence of [gamma-33P]ATP by hotspot kinase assay | Homo sapiens | 2 | ALA5053493 | assay format | Scientific Literature | |
| 11. | ALA5053798 | B | Inhibition of TRKA G595R mutant (unknown origin) in presence of [gamma-33P]ATP by hotspot kinase assay | Homo sapiens | 2 | ALA5053493 | assay format | Scientific Literature | |
| 12. | ALA5053799 | B | Inhibition of TRKA G667C mutant (unknown origin) in presence of [gamma-33P]ATP by hotspot kinase assay | Homo sapiens | 2 | ALA5053493 | assay format | Scientific Literature | |
| 13. | ALA5053800 | B | Inhibition of TRKA L657M mutant (unknown origin) in presence of [gamma-33P]ATP by hotspot kinase assay | Homo sapiens | 2 | ALA5053493 | assay format | Scientific Literature | |
| 14. | ALA5053801 | B | Selectivity index, ratio of IC50 for inhibition of wildtype TRKA (unknown origin) to IC50 for inhibition of TRKA G595R mutant (unknown origin) | Homo sapiens | 6 | ALA5053493 | assay format | Scientific Literature | |
| 15. | ALA5053802 | B | Selectivity index, ratio of IC50 for inhibition of wildtype TRKA (unknown origin) to IC50 for inhibition of TRKA G667C mutant (unknown origin) | Homo sapiens | 6 | ALA5053493 | assay format | Scientific Literature | |
| 16. | ALA5053803 | B | Selectivity index, ratio of IC50 for inhibition of wildtype TRKA (unknown origin) to IC50 for inhibition of TRKA G595R/G667C double mutant (unknown origin) | Homo sapiens | 6 | ALA5053493 | assay format | Scientific Literature | |
| 17. | ALA5053804 | B | Inhibition of wildtype human TRKA using poly (Glu,Tyr) 4:1 as substrate in presence of [gamma-33P]ATP by hotspot kinase assay | Homo sapiens | 6 | ALA5053493 | single protein format | Scientific Literature | |
| 18. | ALA5139763 | B | Inhibition of N-terminal human TRKA (436 to 790 residues) expressed in baculovirus expression system using TK as substrate measured after 30 mins in presence of ATP by HTRF assay | Homo sapiens | 39 | ALA5137027 | assay format | Scientific Literature | |
| 19. | ALA5139764 | B | Inhibition of N-terminal human TRKB (456 to 822 residues) expressed in baculovirus expression system using TK as substrate measured after 40 mins in presence of ATP by HTRF assay | Homo sapiens | 7 | ALA5137027 | assay format | Scientific Literature | |
| 20. | ALA5139765 | B | Inhibition of N-terminal human TRKC (456 to 825 residues) expressed in baculovirus expression system using TK as substrate measured after 40 mins in presence of ATP by HTRF assay | Homo sapiens | 7 | ALA5137027 | assay format | Scientific Literature |
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