| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4818330 | F | Antagonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as inhibition of UDP-induced intracellular calcium mobilization by fluorescence based analysis | Homo sapiens | 26 | ALA4814049 | cell-based format | Scientific Literature | |
| 2. | ALA4818332 | B | Inhibition of alpha2a adrenergic receptor (unknown origin) | Homo sapiens | 6 | ALA4814049 | single protein format | Scientific Literature | |
| 3. | ALA4818333 | B | Inhibition of dopamine D5 receptor (unknown origin) | Homo sapiens | 7 | ALA4814049 | single protein format | Scientific Literature | |
| 4. | ALA4818336 | B | Inhibition of alpha2b adrenergic receptor (unknown origin) | Homo sapiens | 3 | ALA4814049 | single protein format | Scientific Literature | |
| 5. | ALA4818338 | B | Inhibition of dopamine D1 receptor (unknown origin) | Homo sapiens | 1 | ALA4814049 | single protein format | Scientific Literature | |
| 6. | ALA4818339 | B | Inhibition of mu opioid receptor (unknown origin) | Homo sapiens | 1 | ALA4814049 | single protein format | Scientific Literature | |
| 7. | ALA4818340 | B | Inhibition of alpha2c adrenergic receptor (unknown origin) | Homo sapiens | 1 | ALA4814049 | single protein format | Scientific Literature | |
| 8. | ALA5224965 | B | Antagonist activity at Meleagris P2Y1R expressed in human 1321N1 cells assessed as inhibition of UDP-induced calcium mobilization at 100 uM by FLIPR assay relative to control | Meleagris gallopavo | 5 | ALA5223123 | cell-based format | Scientific Literature | |
| 9. | ALA5224966 | B | Antagonist activity at human P2Y2R expressed in human 1321N1 cells assessed as inhibition of UDP-induced calcium mobilization at 100 uM by FLIPR assay relative to control | Homo sapiens | 5 | ALA5223123 | cell-based format | Scientific Literature | |
| 10. | ALA5224967 | B | Antagonist activity at human P2Y4R expressed in human 1321N1 cells assessed as inhibition of UDP-induced calcium mobilization at 100 uM by FLIPR assay relative to control | Homo sapiens | 5 | ALA5223123 | cell-based format | Scientific Literature | |
| 11. | ALA5224969 | B | Antagonist activity at mouse P2Y6R expressed in human 1321N1 cells assessed as inhibition of UDP-induced calcium mobilization at 20 uM by FLIPR assay relative to control | Mus musculus | 2 | ALA5223123 | cell-based format | Scientific Literature | |
| 12. | ALA5224970 | B | Selectivity ratio of IC50 for mouse P2Y6R to IC50 for human P2Y6R | 13 | ALA5223123 | assay format | Scientific Literature | ||
| 13. | ALA5224980 | T | Cytotoxicity against HEK293 cells assessed as reduction in cell viability at 100 uM measured after 24 hrs by MTT assay relative to control | Homo sapiens | 5 | ALA5223123 | cell-based format | Scientific Literature |
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