# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4813853 | B | Inhibition of recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)pLysS cells interaction with FITC-9mer Nrf2 (unknown origin) incubated for 30 mins under shaking condition by fluorescence polarization assay | Homo sapiens | 26 | cell-based format | Scientific Literature | ||
2. | ALA4813854 | B | Inhibition of recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)pLysS cells interaction with FITC-9mer Nrf2 (unknown origin) incubated for 30 mins under shaking condition by TR-FRET assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
3. | ALA4813855 | B | Inhibition of recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)pLysS cells interaction with FITC-9mer Nrf2 (unknown origin) at 50 uM incubated for 30 mins under shaking condition by fluorescence polarization assay relative to control | Homo sapiens | 26 | cell-based format | Scientific Literature | ||
4. | ALA4813856 | B | Inhibition of recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)pLysS cells interaction with FITC-9mer Nrf2 (unknown origin) at 5 uM incubated for 30 mins under shaking condition by fluorescence polarization assay relative to control | Homo sapiens | 26 | cell-based format | Scientific Literature | ||
5. | ALA4813857 | B | Inhibition of recombinant human KEAP1 Kelch domain (321 to 609 residues) expressed in Escherichia coli BL21 (DE3)pLysS cells interaction with FITC-9mer Nrf2 (unknown origin) at 0.5 uM incubated for 30 mins under shaking condition by fluorescence polarization assay relative to control | Homo sapiens | 24 | cell-based format | Scientific Literature | ||
6. | ALA5230560 | B | Binding affinity to human KEAP1 by isothermal titration calorimetric assay | Homo sapiens | 4 | single protein format | Scientific Literature | ||
7. | ALA5230561 | B | Inhibition of human Keap1-Nrf2 protein-protein interaction by fluorescence polarization assay | Homo sapiens | 14 | protein format | Scientific Literature | ||
8. | ALA5230564 | B | Inhibition of human Keap1-Nrf2 protein-protein interaction | Homo sapiens | 1 | protein format | Scientific Literature |