# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4810338 | Binding | Inhibition of human His-ENL YEATS domain and biotinylated H3K9ac peptide interaction by AlphaScreen assay | Homo sapiens | 28 | ALA4808215 | single protein format | Scientific Literature | |
2. | ALA4810340 | Functional | Growth inhibition of ENL-independent human U2OS cells at 50 uM incubated for 3 days by CellTiter-Glo luminescent cell viability assay relative to control | Homo sapiens | 1 | ALA4808215 | cell-based format | Scientific Literature | |
3. | ALA4810341 | Binding | Inhibition of human His-AF9 YEATS domain and biotinylated H3K9ac peptide interaction by AlphaScreen assay | Homo sapiens | 4 | ALA4808215 | single protein format | Scientific Literature | |
4. | ALA4810342 | Binding | Inhibition of human His-GAS41 YEATS domain and biotinylated H3K27ac peptide interaction by AlphaScreen assay | Homo sapiens | 4 | ALA4808215 | single protein format | Scientific Literature | |
5. | ALA4810343 | Binding | Inhibition of human His-YEATS2 YEATS domain and biotinylated H3K27ar peptide interaction by AlphaScreen assay | Homo sapiens | 4 | ALA4808215 | single protein format | Scientific Literature | |
6. | ALA4810345 | Binding | Inhibition of human His-ENL YEATS domain and biotinylated H3K9ac peptide interaction at 5 uM by AlphaScreen assay | Homo sapiens | 2 | ALA4808215 | single protein format | Scientific Literature | |
7. | ALA4810346 | Binding | Inhibition of human His-AF9 YEATS domain and biotinylated H3K9ac peptide interaction at 20 uM by AlphaScreen assay | Homo sapiens | 4 | ALA4808215 | single protein format | Scientific Literature | |
8. | ALA4810347 | Binding | Inhibition of human His-GAS41 YEATS domain and biotinylated H3K27ac peptide interaction at 20 uM by AlphaScreen assay | Homo sapiens | 4 | ALA4808215 | single protein format | Scientific Literature | |
9. | ALA4810348 | Binding | Inhibition of human His-YEATS2 YEATS domain and biotinylated H3K27ar peptide interaction at 20 uM by AlphaScreen assay | Homo sapiens | 4 | ALA4808215 | single protein format | Scientific Literature | |
10. | ALA4810350 | Functional | Growth inhibition of human MOLM13 cells at 5 uM incubated for 3 days by CellTiter-Glo luminescent cell viability assay relative to control | Homo sapiens | 1 | ALA4808215 | cell-based format | Scientific Literature | |
11. | ALA4810351 | Functional | Growth inhibition of human MOLM13 cells at 10 uM incubated for 3 days by CellTiter-Glo luminescent cell viability assay relative to control | Homo sapiens | 1 | ALA4808215 | cell-based format | Scientific Literature | |
12. | ALA4810352 | Functional | Growth inhibition of human MV4-11 cells at 2.5 to 50 uM incubated for 3 days by CellTiter-Glo luminescent cell viability assay relative to control | Homo sapiens | 1 | ALA4808215 | cell-based format | Scientific Literature | |
13. | ALA4810353 | Binding | Stabilization of ENL in human MV4-11 cells assessed as inhibition of high temperature-induced ENL protein degradation at 20 uM incubated for 5 hrs by cellular thermal shift assay | Homo sapiens | 1 | ALA4808215 | cell-based format | Scientific Literature | |
14. | ALA4810354 | Binding | Stabilization of ENL in human MOLM13 cells assessed as inhibition of high temperature-induced ENL protein degradation at 20 uM incubated for 5 hrs by cellular thermal shift assay | Homo sapiens | 1 | ALA4808215 | cell-based format | Scientific Literature | |
15. | ALA4810355 | Binding | Stabilization of GAS41 in human MV4-11 cells assessed as inhibition of high temperature-induced GAS41 protein degradation at 20 uM incubated for 5 hrs by cellular thermal shift assay | Homo sapiens | 1 | ALA4808215 | cell-based format | Scientific Literature | |
16. | ALA4810356 | Binding | Stabilization of GAS41 in human MOLM13 cells assessed as inhibition of high temperature-induced GAS41 protein degradation at 20 uM incubated for 5 hrs by cellular thermal shift assay | Homo sapiens | 1 | ALA4808215 | cell-based format | Scientific Literature | |
17. | ALA4810357 | Binding | Stabilization of ENL in human HeLa cells assessed as inhibition of high temperature-induced ENL protein degradation at 20 uM incubated for 5 hrs by cellular thermal shift assay | Homo sapiens | 1 | ALA4808215 | cell-based format | Scientific Literature | |
18. | ALA4810358 | Binding | Stabilization of AF9 in human HeLa cells assessed as inhibition of high temperature-induced AF9 protein degradation at 20 uM incubated for 5 hrs by cellular thermal shift assay | Homo sapiens | 1 | ALA4808215 | cell-based format | Scientific Literature | |
19. | ALA4810359 | Functional | Growth inhibition of human MOLM-13 cells incubated for 3 days by CellTiter-Glo luminescent cell viability assay | Homo sapiens | 1 | ALA4808215 | cell-based format | Scientific Literature | |
20. | ALA4810360 | Functional | Growth inhibition of human MOLM13 cells incubated for 3 days in presence of JQ1 by CellTiter-Glo luminescent cell viability assay | Homo sapiens | 1 | ALA4808215 | cell-based format | Scientific Literature |