# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4841968 | B | Displacement of [3H]UR-KK200 from human neuropeptide Y Y4 receptor expressed in CHO-mtAEQ cells co-expressing Gqi5 measured after 90 mins by scintillation counting analysis | Homo sapiens | 25 | cell-based format | Scientific Literature | ||
2. | ALA4841969 | B | Displacement of [3H]UR-KK200 from human neuropeptide Y Y4 receptor expressed in CHO-mtAEQ cells co-expressing Gqi5 assessed as fold change in affinity measured after 90 mins by scintillation counting analysis relative to Ac-Arg-Tyr-Arg-Leu-Arg-Tyr-NH2 | Homo sapiens | 19 | cell-based format | Scientific Literature | ||
3. | ALA4841970 | B | Displacement of [3H]UR-MK299 from human neuropeptide Y Y1 receptor in human SK-N-MC cells measured after 90 mins by scintillation counting analysis | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
4. | ALA4841971 | B | Displacement of [3H]UR-MK299 from human neuropeptide Y Y2 receptor expressed in CHO cells measured after 90 mins by scintillation counting analysis | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
5. | ALA4841972 | B | Displacement of [3H]propionyl-pNPY from human neuropeptide Y Y5 receptor in human HEC-1B cells measured after 90 mins by scintillation counting analysis | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
6. | ALA4841973 | B | Selectivity ratio, Ki for displacement of [3H]UR-MK299 from human neuropeptide Y Y1 receptor in human SK-N-MC cells measured after 90 mins by scintillation counting analysis to Ki for displacement of [3H]UR-KK200 from human neuropeptide Y Y4 receptor expressed in CHO-mtAEQ cells co-expressing Gqi5 measured after 90 mins by scintillation counting analysis | Homo sapiens | 18 | cell-based format | Scientific Literature | ||
7. | ALA4841974 | B | Selectivity ratio, Ki for displacement of [3H]UR-MK299 from human neuropeptide Y Y2 receptor expressed in CHO cells measured after 90 mins by scintillation counting analysis to Ki for displacement of [3H]UR-KK200 from human neuropeptide Y Y4 receptor expressed in CHO-mtAEQ cells co-expressing Gqi5 measured after 90 mins by scintillation counting analysis | Homo sapiens | 18 | cell-based format | Scientific Literature | ||
8. | ALA4841975 | B | Selectivity ratio, Ki for displacement of [3H]propionyl-pNPY from human neuropeptide Y Y5 receptor in human HEC-1B cells measured after 90 mins by scintillation counting analysis to Ki for displacement of [3H]UR-KK200 from human neuropeptide Y Y4 receptor expressed in CHO-mtAEQ cells co-expressing Gqi5 measured after 90 mins by scintillation counting analysis | Homo sapiens | 18 | cell-based format | Scientific Literature | ||
9. | ALA4841976 | F | Agonist activity at human neuropeptide Y Y4 receptor expressed in HEK293T-ARRB1 cells assessed as stimulation of beta-arrestin 1 recruitment by multimode plate reader | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
10. | ALA4841977 | F | Intrinsic activity at human neuropeptide Y Y4 receptor expressed in HEK293T-ARRB1 cells assessed as stimulation of beta-arrestin 1 recruitment by multimode plate reader relative to hPP | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
11. | ALA4841978 | F | Agonist activity at human neuropeptide Y Y4 receptor expressed in HEK293T-ARRB2 cells assessed as stimulation of beta-arrestin 2 recruitment by multimode plate reader | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
12. | ALA4841979 | F | Intrinsic activity at human neuropeptide Y Y4 receptor expressed in HEK293T-ARRB2 cells assessed as stimulation of beta-arrestin 2 recruitment by multimode plate reader relative to hPP | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
13. | ALA4841980 | F | Agonist activity at human neuropeptide Y Y4 receptor expressed in CHO-mtAEQ cells co-expressing Gqi5 by calcium aequorin assay | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
14. | ALA4841981 | F | Intrinsic activity at human neuropeptide Y Y4 receptor expressed in CHO-mtAEQ cells co-expressing Gqi5 by calcium aequorin assay | Homo sapiens | 21 | cell-based format | Scientific Literature |