| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4808885 | Binding | Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting method | Homo sapiens | 27 | ALA4808176 | cell membrane format | Scientific Literature | |
| 2. | ALA4808886 | Functional | Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP production | Homo sapiens | 19 | ALA4808176 | cell-based format | Scientific Literature | |
| 3. | ALA4808888 | Functional | Agonist activity at human GCGR expressed in HEK293 cells assessed as stimulation of cAMP production relative to control | Homo sapiens | 10 | ALA4808176 | cell-based format | Scientific Literature | |
| 4. | ALA4808891 | Functional | Antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP production by schild plot analysis | Homo sapiens | 4 | ALA4808176 | cell-based format | Scientific Literature |
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