# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4808885 | Binding | Displacement of 125I-glucagon from human GCGR expressed in HEK293 cells membranes incubated for 6 hrs by liquid scintillation counting method | Homo sapiens | 27 | ALA4808176 | cell membrane format | Scientific Literature | |
2. | ALA4808887 | Functional | Partial antagonist activity at human GCGR expressed in HEK293 cells assessed as inhibition of glucogon-induced cAMP production | Homo sapiens | 8 | ALA4808176 | cell-based format | Scientific Literature | |
3. | ALA4808888 | Functional | Agonist activity at human GCGR expressed in HEK293 cells assessed as stimulation of cAMP production relative to control | Homo sapiens | 10 | ALA4808176 | cell-based format | Scientific Literature |