| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4841800 | Binding | Inhibition of TNNI3K (unknown origin) | Homo sapiens | 53 | ALA4840354 | single protein format | Scientific Literature | |
| 2. | ALA4841801 | Binding | Inhibition of human myc-TNNI3K expressed in HEK-MSR2 cells assessed as reduction in TNNI3K autophosphorylation preincubated for 30 mins followed by pervanadate addition and measured after 20 mins by DELFIA | Homo sapiens | 11 | ALA4840354 | cell-based format | Scientific Literature | |
| 3. | ALA4841802 | Binding | Inhibition of GST-6His tagged VEGFR2 (unknown origin) using biotin-aminohexyl-EEEEYFELVAKKKK-NH2 peptide substrate incubated for 90 mins by HTRF assay | Homo sapiens | 49 | ALA4840354 | single protein format | Scientific Literature | |
| 4. | ALA4841803 | Binding | Inhibition of p38alpha (unknown origin) | Homo sapiens | 50 | ALA4840354 | single protein format | Scientific Literature | |
| 5. | ALA4841804 | Binding | Inhibition of B-Raf (unknown origin) | Homo sapiens | 53 | ALA4840354 | single protein format | Scientific Literature | |
| 6. | ALA4841805 | Binding | Selectivity index, ratio of IC50 for inhibition of VEGFR2 (unknown origin) to IC50 for inhibition of TNNI3K (unknown origin) | Homo sapiens | 49 | ALA4840354 | assay format | Scientific Literature | |
| 7. | ALA4841806 | Binding | Selectivity index, ratio of IC50 for inhibition of p38alpha (unknown origin) to IC50 for inhibition of TNNI3K (unknown origin) | Homo sapiens | 49 | ALA4840354 | assay format | Scientific Literature | |
| 8. | ALA4841807 | Binding | Selectivity index, ratio of IC50 for inhibition of B-Raf (unknown origin) to IC50 for inhibition of TNNI3K (unknown origin) | Homo sapiens | 51 | ALA4840354 | assay format | Scientific Literature | |
| 9. | ALA4841808 | ADME | Permeability of compound incubated for 2 hrs by liquid chromatography analysis | 8 | ALA4840354 | assay format | Scientific Literature | ||
| 10. | ALA4841809 | ADME | Dose normalized AUC in po dosed rat administered as cassette dose | Rattus norvegicus | 11 | ALA4840354 | organism-based format | Scientific Literature | |
| 11. | ALA4841810 | ADME | Half life in po dosed rat administered as cassette dose | Rattus norvegicus | 8 | ALA4840354 | organism-based format | Scientific Literature |
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