| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4836608 | Binding | Inhibition of 6His-Thr-BRD2 (1 to 473 residues) BD1 domain (unknown origin) incubated for 30 mins by TR-FRET assay | Homo sapiens | 1 | ALA4834466 | single protein format | Scientific Literature | |
| 2. | ALA4836609 | Binding | Selectivity index, ratio of pIC50 of recombinant human BRDT BD2 (250 to 382 residues) expressed in bacterial expression system to pIC50 of recombinant human BRDT BD1 (21 to 137 residues) expressed in bacterial expression system | Homo sapiens | 1 | ALA4834466 | assay format | Scientific Literature | |
| 3. | ALA4836610 | Binding | Selectivity index, ratio of pIC50 of recombinant human BRD4 BD2 (333 to 460 residues) expressed in bacterial expression system to pIC50 of recombinant human BRD4 BD1 (44 to 168 residues) expressed in bacterial expression system | Homo sapiens | 1 | ALA4834466 | assay format | Scientific Literature | |
| 4. | ALA4836611 | Binding | Selectivity index, ratio of pIC50 of recombinant human BRD3 BD2 (306 to 416 residues) expressed in bacterial expression system to pIC50 of recombinant human BRD3 BD1 (24 to 144 residues) expressed in bacterial expression system | Homo sapiens | 1 | ALA4834466 | assay format | Scientific Literature | |
| 5. | ALA4836612 | Binding | Selectivity index, ratio of pIC50 of recombinant human BRD2 BD2 (348 to 455 residues) expressed in bacterial expression system to pIC50 of recombinant human BRD2 BD1 (71 to 194 residues) expressed in bacterial expression system | Homo sapiens | 1 | ALA4834466 | assay format | Scientific Literature | |
| 6. | ALA4836613 | Binding | Inhibition of recombinant human BRDT BD2 (250 to 382 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 1 | ALA4834466 | assay format | Scientific Literature | |
| 7. | ALA4836614 | Binding | Inhibition of recombinant human BRDT BD1 (21 to 137 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 1 | ALA4834466 | assay format | Scientific Literature | |
| 8. | ALA4836615 | Binding | Inhibition of recombinant human BRD4 BD2 (333 to 460 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 1 | ALA4834466 | assay format | Scientific Literature | |
| 9. | ALA4836616 | Binding | Inhibition of recombinant human BRD4 BD1 (44 to 168 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 1 | ALA4834466 | assay format | Scientific Literature | |
| 10. | ALA4836617 | Binding | Inhibition of recombinant human BRD3 BD2 (306 to 416 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 1 | ALA4834466 | assay format | Scientific Literature | |
| 11. | ALA4836618 | Binding | Inhibition of recombinant human BRD2 BD2 (348 to 455 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 1 | ALA4834466 | assay format | Scientific Literature | |
| 12. | ALA4836619 | Binding | Inhibition of recombinant human BRD3 BD1 (24 to 144 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 1 | ALA4834466 | assay format | Scientific Literature | |
| 13. | ALA4836620 | Binding | Inhibition of recombinant human BRD2 BD1 (71 to 194 residues) expressed in bacterial expression system by bromoscan assay | Homo sapiens | 1 | ALA4834466 | assay format | Scientific Literature | |
| 14. | ALA4836621 | Binding | Selectivity index, ratio of pIC50 of 6His-FLAG-Tev-BRDT (1 to 397 residues) BD2 domain Y309A or Y66A mutant (unknown origin) to pIC50 of 6His-FLAG-Tev-BRDT (1 to 397 residues) BD1 domain (unknown origin) | Homo sapiens | 1 | ALA4834466 | assay format | Scientific Literature | |
| 15. | ALA4836622 | Binding | Selectivity index, ratio of pIC50 of 6His-Thr-BRD3 (1 to 435 residues) BD2 domain Y348A or Y73A mutant (unknown origin) to pIC50 of 6His-Thr-BRD3 (1 to 435 residues) BD1 domain (unknown origin) | Homo sapiens | 1 | ALA4834466 | assay format | Scientific Literature | |
| 16. | ALA4836623 | Binding | Inhibition of 6His-FLAG-Tev-BRDT (1 to 397 residues) BD1 domain (unknown origin) incubated for 30 mins by TR-FRET assay | Homo sapiens | 1 | ALA4834466 | single protein format | Scientific Literature | |
| 17. | ALA4836624 | Binding | Selectivity index, ratio of pIC50 of 6His-Thr-BRD2 (1 to 473 residues) BD2 domain Y386A or Y113A mutant (unknown origin) to pIC50 of 6His-Thr-BRD2 (1 to 473 residues) BD1 domain (unknown origin) | Homo sapiens | 1 | ALA4834466 | assay format | Scientific Literature | |
| 18. | ALA4836625 | Binding | Inhibition of 6His-FLAG-Tev-BRDT (1 to 397 residues) BD2 domain Y309A or Y66A mutant (unknown origin) incubated for 30 mins by TR-FRET assay | Homo sapiens | 1 | ALA4834466 | single protein format | Scientific Literature | |
| 19. | ALA4836626 | Binding | Inhibition of 6His-Thr-BRD3 (1 to 435 residues) BD1 domain (unknown origin) incubated for 30 mins by TR-FRET assay | Homo sapiens | 1 | ALA4834466 | single protein format | Scientific Literature | |
| 20. | ALA4836627 | Binding | Inhibition of 6His-Thr-BRD3 (1 to 435 residues) BD2 domain Y348A or Y73A mutant (unknown origin) incubated for 30 mins by TR-FRET assay | Homo sapiens | 1 | ALA4834466 | single protein format | Scientific Literature |
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