| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4824071 | Binding | Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assay | Homo sapiens | 35 | ALA4823258 | single protein format | Scientific Literature | |
| 2. | ALA4824072 | Binding | Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assay | Homo sapiens | 35 | ALA4823258 | single protein format | Scientific Literature | |
| 3. | ALA4824073 | Binding | Selectivity ratio of IC50 for His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate to IC50 for His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assay | Homo sapiens | 35 | ALA4823258 | assay format | Scientific Literature | |
| 4. | ALA4824074 | Binding | Binding affinity to human partial length CREBBP (R1081 to G1197 residues) expressed in bacterial expression system assessed as melting temperature by differential scanning fluorometry (Rvb = 46.7 degreeC) | Homo sapiens | 4 | ALA4823258 | assay format | Scientific Literature | |
| 5. | ALA4824075 | Binding | Binding affinity to human partial length EP300 (A1040 to G1161 residues) expressed in bacterial expression system assessed as melting temperature by differential scanning fluorometry (Rvb = 42.1 degreeC) | Homo sapiens | 4 | ALA4823258 | assay format | Scientific Literature | |
| 6. | ALA4824076 | Binding | Binding affinity to human partial length BRD4 bromodomain 1 long isoform (N44 to E168 residues) expressed in bacterial expression system assessed as melting temperature by differential scanning fluorometry (Rvb = 50.1 degreeC) | Homo sapiens | 4 | ALA4823258 | assay format | Scientific Literature |
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