| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4832170 | B | Inhibition of human recombinant MAGL using 4-NPA as substrate by microplate reader method | Homo sapiens | 20 | single protein format | Scientific Literature | ||
| 2. | ALA4832171 | B | Inhibition of human recombinant MAGL in presence of 10 uM DTT for 15 mins by DTT interference assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 3. | ALA4832172 | B | Reversible inhibition of human recombinant MAGL at 320 nM pre-incubated for 60 mins before 4-NPA substrate addition by dilution assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 4. | ALA4832173 | B | Reversible inhibition of human recombinant MAGL at 8 nM pre-incubated for 60 mins before 4-NPA substrate addition by dilution assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 5. | ALA4832174 | B | Reversible inhibition of human recombinant MAGL pre-incubated upto 60 mins before 4-NPA substrate addition by preincubation assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 6. | ALA4832175 | B | Inhibition of human recombinant MAGL assessed as dissociation constant using 4-NPA as substrate | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 7. | ALA4832176 | B | Inhibition of human recombinant FAAH using AMC arachidonoyl amyl as substrate by fluorescence based assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 8. | ALA4832177 | F | Antiproliferative activity against human COLO201 cells assessed as inhibition of cell viability for 96 hrs by cell titre glo luminescence assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 9. | ALA4832178 | F | Antiproliferative activity against human COLO205 cells assessed as inhibition of cell viability for 96 hrs by cell titre glo luminescence assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 10. | ALA4832179 | F | Antiproliferative activity against human HCT-116 cells assessed as inhibition of cell viability for 96 hrs by cell titre glo luminescence assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 11. | ALA4832180 | F | Antiproliferative activity against human HT-29 cells assessed as inhibition of cell viability for 96 hrs by cell titre glo luminescence assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 12. | ALA4832181 | F | Antiproliferative activity against human KURAMOCHI cells assessed as inhibition of cell viability for 96 hrs by cell titre glo luminescence assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 13. | ALA4832182 | F | Antiproliferative activity against human OVCAR-3 cells assessed as inhibition of cell viability for 96 hrs by cell titre glo luminescence assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 14. | ALA4832183 | F | Antiproliferative activity against human OVCAR-5 cells assessed as inhibition of cell viability for 96 hrs by cell titre glo luminescence assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 15. | ALA4832184 | F | Antiproliferative activity against human SK-OV-3 cells assessed as inhibition of cell viability for 96 hrs by cell titre glo luminescence assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 16. | ALA4832185 | F | Antiproliferative activity against human MDA-MB-231 cells assessed as inhibition of cell viability for 96 hrs by cell titre glo luminescence assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 17. | ALA5166863 | A | Stability of the compound in pooled human plasma at 3 mM measured up to 24 hrs by UV/LC-MS assay | Homo sapiens | 2 | cell-free format | Scientific Literature | ||
| 18. | ALA5166864 | A | Metabolic stability in human liver microsomes incubated for 1 hr in presence of NADPH regenerating system by UV/LC-MS analysis | Homo sapiens | 2 | microsome format | Scientific Literature | ||
| 19. | ALA5166865 | P | Stability of the compound in MeOH solution at 500 uM measured up to 24 hrs by UV/LC-MS analysis | 2 | small-molecule physicochemical format | Scientific Literature | |||
| 20. | ALA5166869 | A | Apparent permeability of the compound in PBS buffer pH 7.4 assessed as membrane retention at 0.5 mM incubated for 5 hrs by PAMPA based UV/LC-MS analysis | 2 | assay format | Scientific Literature |
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