| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4825222 | Binding | Inhibition of N-terminal GST-tagged human recombinant C-KIT V654A mutant (544 to end residues) using GGMEDIYEFMGGKKK as substrate measured after 40 mins in presence of [gamma-33P]ATP by scintillation counting analysis | Homo sapiens | 12 | ALA4823309 | single protein format | Scientific Literature | |
| 2. | ALA4825223 | Binding | Inhibition of C-KIT V654A/560-576 deletion mutant in human GIST-430/654 cells assessed as reduction in c-Kit autophosphorylation at Tyr307 residue incubated for 45 mins by Luminex bead based assay | Homo sapiens | 12 | ALA4823309 | cell-based format | Scientific Literature |
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