| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4838928 | B | Inhibition of human proteasome subunit beta-5i chymotrypsin like activity using SUC-ANW-AMC as flurogenic substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by fluorescence assay | Homo sapiens | 21 | single protein format | Scientific Literature | ||
| 2. | ALA4838929 | B | Inhibition of chymotrypsin-like activity of human 20s proteasome beta 5c subunit using suc-WLA-AMC as flurogenic substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by fluorescence assay | Homo sapiens | 21 | single protein format | Scientific Literature | ||
| 3. | ALA4838930 | B | Inhibition of caspase-like activity of human proteasome beta-1c subunit using SUC-LLE-AMC as flurogenic substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by fluorescence assay | Homo sapiens | 6 | single protein format | Scientific Literature | ||
| 4. | ALA4838931 | B | Inhibition of human caspase-like activity of 20s proteasome beta 1i subunit using SUC-PAL-AMC as flurogenic substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by fluorescence assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 5. | ALA4838932 | B | Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by fluorescence assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 6. | ALA4838933 | B | Inhibition of human trypsin-like activity of 20s proteasome beta 2i subunit using SUC-VGR-AMC as flurogenic substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by fluorescence assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 7. | ALA4838934 | B | Selectivity ratio of IC50 for chymotrypsin-like activity of human 20s proteasome beta 5c subunit to IC50 for human proteasome subunit beta-5i chymotrypsin like activity | 21 | assay format | Scientific Literature | |||
| 8. | ALA4838935 | F | Antiproliferative activity against human RPMI-8226 cells assessed as inhibition of cell proliferation after 72 hrs by MTS assay | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 9. | ALA4838936 | F | Antiproliferative activity against human MM1.S cells assessed as inhibition of cell proliferation after 72 hrs by MTS assay | Homo sapiens | 5 | cell-based format | Scientific Literature |
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