| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4829967 | B | Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by HTRF assay | Homo sapiens | 17 | cell-based format | Scientific Literature | ||
| 2. | ALA4829969 | B | Binding affinity to N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells by SPR assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 3. | ALA4829970 | B | Binding affinity to N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells at 200 uM by CPMG NMR spectroscopy | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 4. | ALA4829971 | B | Binding affinity to N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells at 200 uM by STD NMR spectroscopy | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 5. | ALA4829972 | B | Inhibition of BRD2-BD1 (unknown origin) at 1 uM using acetylated H4 as substrate incubated for 1 hr by AlphaScreen assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA4829973 | B | Inhibition of BRD2-BD2 (unknown origin) at 1 uM using acetylated H4 as substrate incubated for 1 hr by AlphaScreen assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 7. | ALA4829974 | B | Inhibition of BRD4-BD1 (unknown origin) at 1 uM using acetylated H4 as substrate incubated for 1 hr by AlphaScreen assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA4829975 | B | Inhibition of BRD4-BD2 (unknown origin) at 1 uM using acetylated H4 as substrate incubated for 1 hr by AlphaScreen assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA4829976 | B | Inhibition of p300-BRD (unknown origin) at 1 uM using acetylated H4 as substrate incubated for 1 hr by AlphaScreen assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA4829977 | B | Inhibition of CBP-BRD (unknown origin) at 1 uM using acetylated H4 as substrate incubated for 1 hr by AlphaScreen assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA4829978 | B | Inhibition of SMARCA2-BRD (unknown origin) at 1 uM using acetylated H4 as substrate incubated for 1 hr by AlphaScreen assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA4829979 | B | Inhibition of N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells at 1 uM incubated for 1 hr by AlphaScreen assay relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 13. | ALA4829980 | B | Binding affinity to N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells assessed as change in melting temperature at 25 uM by thermal shift assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 14. | ALA4829981 | B | Binding affinity to N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells assessed as change in melting temperature at 50 uM by thermal shift assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 15. | ALA4829982 | B | Binding affinity to N-terminal GST-tagged human BPTF (2914 to 3037 residues) expressed in Escherichia coli BL21-CodonPlus (DE3) cells assessed as change in melting temperature at 100 uM by thermal shift assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 16. | ALA4829983 | B | Binding affinity to BRD4-BD1 (unknown origin) assessed as change in melting temperature at 50 uM by thermal shift assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA4829984 | B | Binding affinity to BRD4-BD2 (unknown origin) assessed as change in melting temperature at 50 uM by thermal shift assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA4829985 | B | Binding affinity to BRD2-BD1 (unknown origin) assessed as change in melting temperature at 50 uM by thermal shift assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA4829986 | B | Binding affinity to BRD2-BD2 (unknown origin) assessed as change in melting temperature at 50 uM by thermal shift assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 20. | ALA4829987 | B | Binding affinity to SMARCA2-BRD (unknown origin) assessed as change in melting temperature at 50 uM by thermal shift assay | Homo sapiens | 1 | single protein format | Scientific Literature |
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