| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4812854 | Binding | Displacement of [125-I]-[Sar1, Ile8] from recombinant human AT1R transfected in human HEK293 cells incubated for 2 hrs by liquid scintillation counter analysis | Homo sapiens | 10 | ALA4811266 | cell-based format | Scientific Literature | |
| 2. | ALA4812855 | Binding | Displacement of [125-I]-[Sar1, Ile8] from recombinant human AT2R transfected in human HEK293 cells incubated for 2 hrs by liquid scintillation counter analysis | Homo sapiens | 10 | ALA4811266 | cell-based format | Scientific Literature | |
| 3. | ALA4812856 | Binding | Selectivity index, ratio of IC50 for displacement of [125-I]-[Sar1, Ile8] from recombinant human AT2R transfected in human HEK293 cells to IC50 for displacement of [125-I]-[Sar1, Ile8] from recombinant human AT1R transfected in human HEK293 cells | Homo sapiens | 10 | ALA4811266 | cell-based format | Scientific Literature | |
| 4. | ALA4812857 | ADME | Stability of compound in human plasma assessed as parent compound remaining incubated for 24 hrs by LC-MS/MS analysis | Homo sapiens | 9 | ALA4811266 | cell-free format | Scientific Literature |
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