# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA4819715 | Binding | Binding affinity to wild-type human partial length TTK (N505 to V798 residues) expressed in bacterial expression system by active site-directed competition binding based Kinomescan method | Homo sapiens | 30 | ALA4818999 | assay format | Scientific Literature | |
2. | ALA4819716 | Binding | Inhibition of recombinant full-length human TTK using MBP as substrate incubated for 40 mins in presence of [gamma33P]ATP by scintillation counting based radiometry assay relative to control | Homo sapiens | 6 | ALA4818999 | single protein format | Scientific Literature | |
3. | ALA4819717 | Binding | Inhibition of recombinant full-length human TTK at 100 nM using MBP as substrate incubated for 40 mins in presence of [gamma33P]ATP by scintillation counting based radiometry assay relative to control | Homo sapiens | 1 | ALA4818999 | single protein format | Scientific Literature | |
4. | ALA4819718 | Binding | Binding affinity to wild-type human partial length PIK3CD (R108 to Q1044 residues) expressed in HEK293 cells by active site-directed competition binding based Kinomescan method | Homo sapiens | 1 | ALA4818999 | cell-based format | Scientific Literature | |
5. | ALA4819719 | Binding | Binding affinity to wild-type human partial length DAPK3 (M1 to A277 residues) expressed in bacterial expression system by measuring active site-directed competition binding based Kinomescan method | Homo sapiens | 1 | ALA4818999 | assay format | Scientific Literature | |
6. | ALA4819720 | Binding | Binding affinity to wild-type human full length MARK3 (M1 to L729 residues) expressed in bacterial expression system by measuring active site-directed competition binding based Kinomescan method | Homo sapiens | 1 | ALA4818999 | assay format | Scientific Literature | |
7. | ALA4819721 | Binding | Binding affinity to human partial length PIK3C2G (M1 to I1446 residues) expressed in mammalian expression system by active site-directed competition binding based Kinomescan method | Homo sapiens | 1 | ALA4818999 | assay format | Scientific Literature | |
8. | ALA4819722 | Binding | Binding affinity to wild-type human partial length IRAK1 (R194 to S712 residues) expressed in mammalian expression system by active site-directed competition binding based Kinomescan method | Homo sapiens | 1 | ALA4818999 | assay format | Scientific Literature | |
9. | ALA4819723 | Binding | Inhibition of human PIK3CD at 100 nM by scintillation counting based direct-filter Binding radiometric assay relative to control | Homo sapiens | 1 | ALA4818999 | single protein format | Scientific Literature | |
10. | ALA4819724 | Binding | Inhibition of human DAPK3 at 100 nM by direct-filter Binding radiometric assay relative to control | Homo sapiens | 1 | ALA4818999 | single protein format | Scientific Literature | |
11. | ALA4819725 | Binding | Inhibition of human MARK3 using KKKVSRSGLYRSPSMPENLNRPR as substrate at 100 nM by direct-filter Binding radiometric assay relative to control | Homo sapiens | 1 | ALA4818999 | single protein format | Scientific Literature | |
12. | ALA4819726 | Binding | Inhibition of human full length JNK3 at 100 nM by direct-filter Binding radiometric assay relative to control | Homo sapiens | 1 | ALA4818999 | single protein format | Scientific Literature | |
13. | ALA4819727 | Binding | Inhibition of human STK16 at 100 nM by direct-filter Binding radiometric assay relative to control | Homo sapiens | 1 | ALA4818999 | single protein format | Scientific Literature | |
14. | ALA4819728 | Binding | Inhibition of wild-type human partial length DAPK1 (M1 to F296 residues) using KKLNRTLSFAEPG peptide as substrate at 100 nM by direct-filter Binding radiometric assay relative to control | Homo sapiens | 1 | ALA4818999 | single protein format | Scientific Literature | |
15. | ALA4819729 | Binding | Inhibition of human SNARK assessed as residual activity using KKKVSRSGLYRSPSMPENLNRPR as substrate at 100 nM by direct-filter Binding radiometric assay relative to control | Homo sapiens | 1 | ALA4818999 | single protein format | Scientific Literature | |
16. | ALA4819730 | Binding | Inhibition of human DCAMKL1 at 100 nM by direct-filter Binding radiometric assay relative to control | Homo sapiens | 1 | ALA4818999 | single protein format | Scientific Literature | |
17. | ALA4819731 | Binding | Inhibition of human recombinant MELK (1 to 340 residues) using KKLNRTLSFAEPG peptide as substrate at 100 nM by direct-filter Binding radiometric assay relative to control | Homo sapiens | 1 | ALA4818999 | single protein format | Scientific Literature | |
18. | ALA4819732 | Binding | Inhibition of human STK39 at 100 nM by direct-filter Binding radiometric assay relative t | Homo sapiens | 1 | ALA4818999 | single protein format | Scientific Literature | |
19. | ALA4819733 | Binding | Inhibition of human recombinant full length CSNK2A1 using RRRDDDSDDD peptide as substrate at 100 nM direct filter-binding radiometric kinase activity assay relative to control | Homo sapiens | 1 | ALA4818999 | single protein format | Scientific Literature | |
20. | ALA4819734 | Binding | Inhibition of human recombinant full length DAPK2 using Calmodulin as substrate at 100 nM direct filter-binding radiometric kinase activity assay relative to control | Homo sapiens | 1 | ALA4818999 | single protein format | Scientific Literature |