| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA4810421 | B | Inhibition of recombinant full-length human GRK6 using casein as substrate measured after 80 mins in presence of [gamma33P]ATP by radiometric scintillation counting method | Homo sapiens | 39 | single protein format | Scientific Literature | ||
| 2. | ALA4810423 | B | Inhibition of recombinant full length human Aurora A using LRRASLG as substrate incubated for 40 mins in presence of [gamma-33ATP] by radiometric scintillation counting method | Homo sapiens | 17 | single protein format | Scientific Literature | ||
| 3. | ALA4810424 | B | Inhibition of recombinant human IGF-1R (959 to end residues) using KKKSPGEYVNIEF as substrate incubated for 40 mins in presence of [gamma-33ATP] by radiometric scintillation counting method | Homo sapiens | 9 | single protein format | Scientific Literature | ||
| 4. | ALA4810446 | B | Binding affinity to FLAG-tagged GRK6 in human KMS11 cells incubated for 2.5 hrs by ITDR assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 5. | ALA4810447 | B | Binding affinity to FLAG-tagged GRK6 in human KMS11 cells assessed as half life of GRK6 occupancy at 5 uM preincubated for 2.5 hrs followed by compound washout by ITDR assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 6. | ALA4810448 | B | Selectivity index, ratio of IC50 for inhibition of human Aurora A to IC50 for inhibition of human GRK6 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 7. | ALA4810449 | B | Selectivity index, ratio of IC50 for inhibition of human IGF-1R to IC50 for inhibition of human GRK6 | Homo sapiens | 1 | assay format | Scientific Literature |
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